SCHEMBL4431098

SCHEMBL4431098

CCCCOc1ccc(CC(=O)N(c2ncccc2C#N)C2CCNCC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.37
MAPKAPK2 P49137 1/20 0.37
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
PDE4A P27815 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HIF1A Q16665 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
ITGB3 P05106 6/20 0.36
ITGA2B P08514 6/20 0.36
RPLP1 P05386 2/20 0.36
RPLP0 P05388 2/20 0.36
RPS17 P08708 2/20 0.36
RPSA P08865 2/20 0.36
RPS2 P15880 2/20 0.36
RPL35A P18077 2/20 0.36
RPL7 P18124 2/20 0.36
RPL17 P18621 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3335575 0.78 HRH2 (0.41) HTR2ASMN1; SMN2
SCHEMBL8169931 0.73 JAK2 (0.41) HTR2ACYP2D6SMN1; SMN2NPC1
SCHEMBL3334782 0.70 CYP3A4 (0.44) CYP2D6SMN1; SMN2NOS2NPC1
SCHEMBL3334079 0.69 KDM4E (0.58) HTR2AKDM4ESMN1; SMN2
SCHEMBL8169539 0.69 JAK2 (0.50) SLC6A4NOS2
SCHEMBL3331527 0.69 MEN1 (0.55) HTR2AKDM4ESMN1; SMN2
SCHEMBL11448021 0.66 CHRM3 (0.52) KDM4ECYP2D6SMN1; SMN2KCNH2CHRM2
SCHEMBL3947609 0.66 HTR2A (0.56) HTR2AKCNH2SLC6A4
SCHEMBL3338157 0.66 KDM4E (0.58) HTR2AKDM4ESMN1; SMN2
SCHEMBL22878508 0.65 SLC6A2 (0.47) CYP2D6SMN1; SMN2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134687-A1 PIPERAZINE AND PIPERIDINE MGLUR5 POTENTIATORS AstraZeneca AB (SE) 2009-12-23 EP claimed
WO-2008112440-A1 PIPERAZINE AND PIPERIDINE MGLUR5 POTENTIATORS ASTRAZENECA AB (SE) 2008-09-18 WO claimed