SCHEMBL4432707

SCHEMBL4432707

ClC1=[C]Cc2cccc(Cl)c2N1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.50
HTR5A P47898 1/20 0.47
NSD2 O96028 1/20 0.35
BCHE P06276 1/20 0.35
DAO P14920 1/20 0.35
CES1 P23141 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
PNMT P11086 1/20 0.34
MAPT P10636 1/20 0.33
PDE7A Q13946 1/20 0.32
PDE7B Q9NP56 1/20 0.32
ADRA2A P08913 1/20 0.31
CYP2D6 P10635 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4152022 0.69 AHR (0.42) AHRHTR5ANSD2BCHEDAO
SCHEMBL1162926 0.67 AHR (1.00) AHRHTR5ANSD2BCHEDAO
SCHEMBL1764695 0.65 AHR (0.70) AHRHTR5ANSD2BCHEDAO
SCHEMBL11534863 0.65 AHR (0.59) AHRHTR5ANSD2BCHEDAO
SCHEMBL25369916 0.64 AHR (0.49) AHRHTR5ANSD2BCHEDAO
SCHEMBL30528633 0.64 AHR (0.49) AHRHTR5ANSD2BCHEDAO
SCHEMBL11708913 0.63 AHR (0.47) AHRHTR5ANSD2BCHEDAO
SCHEMBL3284838 0.62 AHR (0.86) AHRHTR5ANSD2BCHEDAO
SCHEMBL31430300 0.62 AHR (0.54) AHRHTR5ANSD2BCHEDAO
SCHEMBL3878574 0.61 MAPT (0.56) AHRHTR5APNMTMAPTADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137186-A1 HETEROCYCLIC COMPOUNDS AND THEIR USES Amgen Inc. (US) 2009-12-30 EP disclosed
WO-2008118468-A1 HETEROCYCLIC COMPOUNDS AND THEIR USES AMGEN INC. (US) 2008-10-02 WO disclosed