SCHEMBL4433065

SCHEMBL4433065

[CH2]c1ccc(C(=O)Nc2cc(-c3ccccc3)ccc2N)cc1

nearest known ligand 0.81

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 15/20 0.81
HDAC1 Q13547 10/20 0.81
HDAC3 O15379 4/20 0.81

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16380794 0.90 HDAC2 (1.00) HDAC2HDAC1HDAC3
SCHEMBL26775695 0.89 HDAC2 (0.86) HDAC2HDAC1HDAC3
SCHEMBL4581182 0.87 HDAC2 (0.83) HDAC2HDAC1HDAC3
SCHEMBL15398029 0.85 HDAC1 (0.81) HDAC2HDAC1HDAC3
SCHEMBL4322002 0.84 HDAC2 (0.77) HDAC2HDAC1HDAC3
SCHEMBL4580508 0.84 HDAC1 (0.77) HDAC2HDAC1HDAC3
SCHEMBL15397970 0.83 HDAC2 (0.86) HDAC2HDAC1HDAC3
SCHEMBL4311556 0.83 HDAC2 (0.75) HDAC2HDAC1HDAC3
SCHEMBL18653511 0.83 HDAC2 (0.75) HDAC2HDAC1HDAC3
SCHEMBL2209647 0.83 HDAC2 (0.75) HDAC2HDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049124-A2 PHOSPHORUS DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS Merck & Co., Inc. (US) 2009-04-22 EP disclosed
WO-2008010985-A2 PHOSPHORUS DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2008-01-24 WO disclosed