SCHEMBL4442280

SCHEMBL4442280

NC(=O)C(F)[C@@]1(C(=O)O)C[C@@H]1c1ccc(-c2ccc(F)cc2)nc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
PTPN1 P18031 1/20 0.37
PTPN6 P29350 1/20 0.37
PTPN11 Q06124 1/20 0.37
KDM1A O60341 9/20 0.36
MAOB P27338 2/20 0.34
LDHA P00338 1/20 0.34
GRIA2 P42262 1/20 0.34
DGAT1 O75907 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
KCNH2 Q12809 1/20 0.33
HTR4 Q13639 1/20 0.33
HDAC2 Q92769 2/20 0.32
TGFBR1 P36897 1/20 0.32
HDAC1 Q13547 1/20 0.32
HPGDS O60760 1/20 0.32
MLNR O43193 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4605637 1.00 NPC1 (0.40) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL4442040 0.76 NPC1 (0.40) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL4449737 0.76 NPC1 (0.40) NPC1RXFP1PTPN1PTPN6PTPN11
Hydrochloric Acid SCHEMBL3605048 0.75 NPC1 (0.45) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL3610730 0.70 NPC1 (0.39) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL3646654 0.69 KDM1A (0.51) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL3646653 0.69 KDM1A (0.51) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL3600203 0.67 KDM1A (0.49) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL3605976 0.67 KDM1A (0.49) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL3600206 0.67 KDM1A (0.49) NPC1RXFP1PTPN1PTPN6PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121612-A1 HETEROARYLCYCLOPROPANECARBOXAMIDES AND THEIR USE AS PHARMACEUTICALS Sanofi-Aventis (FR) 2009-11-25 EP disclosed
WO-2008080511-A1 HETEROARYLCYCLOPROPANECARBOXAMIDES AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (FR) 2008-07-10 WO disclosed