SCHEMBL4443009

SCHEMBL4443009

O=C(O)C1CN(Cc2ccc(-c3cc4cc(CCc5ccccc5)ccc4o3)c(F)c2)C1

nearest known ligand 0.85

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 19/20 0.85
S1PR3 Q99500 9/20 0.85
KCNH2 Q12809 1/20 0.85
S1PR5 Q9H228 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4440616 0.96 S1PR1 (0.82) S1PR1S1PR3KCNH2S1PR5
SCHEMBL1601733 0.92 S1PR1 (1.00) S1PR1S1PR3KCNH2
SCHEMBL4449544 0.91 S1PR1 (0.71) S1PR1S1PR3KCNH2S1PR5
SCHEMBL1601432 0.89 S1PR1 (0.80) S1PR1S1PR3KCNH2S1PR5
SCHEMBL1601562 0.88 S1PR1 (0.88) S1PR1S1PR3KCNH2
SCHEMBL1602925 0.88 S1PR1 (0.84) S1PR1S1PR3KCNH2
SCHEMBL4446551 0.88 S1PR1 (0.69) S1PR1S1PR3KCNH2S1PR5
SCHEMBL1603279 0.87 S1PR1 (0.77) S1PR1S1PR3KCNH2S1PR5
SCHEMBL1602502 0.87 S1PR1 (0.76) S1PR1S1PR3KCNH2
SCHEMBL3696584 0.87 S1PR1 (0.82) S1PR1S1PR3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121648-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX Pharmaceuticals, Inc. (US) 2009-11-25 EP disclosed
WO-2007109334-A2 SIP RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX DELAWARE, INC. (US) 2007-09-27 WO disclosed