SCHEMBL4447764

SCHEMBL4447764

CCOC(=O)c1cccc(-n2nc(C(C)(C)C)cc2NC(=O)Nc2ccc(Oc3ccnc(C(=O)NC)c3)cc2Cl)c1.CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3cc(C(C)C)nn3-c3cc(Cl)cc(Cl)c3)c(F)c2)ccn1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 13/20 0.59
MAPK14 Q16539 7/20 0.59
ABL1 P00519 4/20 0.59
RIPK1 Q13546 2/20 0.59
RAF1 P04049 2/20 0.59
RET P07949 2/20 0.59
KIT P10721 2/20 0.59
BCR P11274 2/20 0.59
FGFR1 P11362 2/20 0.59
PDGFRA P16234 2/20 0.59
FLT1 P17948 2/20 0.59
EPHA1 P21709 2/20 0.59
TTK P33981 2/20 0.59
FLT4 P35916 2/20 0.59
KDR P35968 2/20 0.59
FLT3 P36888 2/20 0.59
MAPKAPK2 P49137 2/20 0.59
CLK1 P49759 2/20 0.59
LIMK1 P53667 2/20 0.59
CDK17 Q00537 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL400258 0.91 BRAF (0.70) BRAFMAPK14ABL1RIPK1RAF1
SCHEMBL2245567 0.91 MAPK14 (0.60) BRAFMAPK14ABL1RIPK1RAF1
SCHEMBL2250309 0.89 MAPK14 (0.57) BRAFMAPK14ABL1RIPK1RAF1
SCHEMBL2240803 0.84 MAPK14 (0.66) BRAFMAPK14ABL1RIPK1RAF1
SCHEMBL1129422 0.84 BRAF (0.74) BRAFMAPK14ABL1RIPK1RAF1
SCHEMBL2241987 0.84 ABL1 (0.78) BRAFMAPK14ABL1RIPK1RAF1
SCHEMBL1129786 0.84 BRAF (0.71) BRAFMAPK14ABL1RIPK1RAF1
SCHEMBL2243621 0.83 MAPK14 (0.52) BRAFMAPK14ABL1RIPK1RAF1
SCHEMBL2241256 0.83 ABL1 (0.62) BRAFMAPK14ABL1RIPK1RAF1
SCHEMBL2242931 0.83 MAPK14 (0.68) BRAFMAPK14ABL1RIPK1RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044053-A2 UREA COMPOUNDS USEFUL IN THE TREATMENT OF CANCER Bayer Healthcare, LLC (US) 2009-04-08 EP claimed
WO-2007064872-A2 UREA COMPOUNDS USEFUL IN THE TREATMENT OF CANCER BAYER HEALTHCARE LLC (US) 2007-06-07 WO claimed