SCHEMBL4448045

SCHEMBL4448045

O=C(OC(=O)c1cc(C=Cc2ccc(C(F)(F)F)c(Cl)c2)ccc1NC(=O)C1CC1)c1cc(C=Cc2ccc(Cl)c(F)c2)ccc1NC(=O)C1CC1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.42
KDR P35968 12/20 0.41
BRAF P15056 7/20 0.40
KCNA3 P22001 1/20 0.38
MEN1 O00255 1/20 0.38
TSHR P16473 1/20 0.38
DHODH Q02127 1/20 0.37
MGLL Q99685 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4448040 0.91 KMT2A (0.43) KMT2AKDRBRAFKCNA3MEN1
SCHEMBL4448047 0.91 KMT2A (0.43) KMT2AKDRBRAFKCNA3MEN1
SCHEMBL1823180 0.85 KMT2A (0.43) KMT2AKDRMEN1TSHRDHODH
SCHEMBL1822975 0.85 KMT2A (0.43) KMT2AKDRMEN1TSHRDHODH
SCHEMBL1822942 0.82 KMT2A (0.51) KMT2AKCNA3MEN1DHODHMGLL
SCHEMBL1822945 0.82 KMT2A (0.51) KMT2AKCNA3MEN1DHODHMGLL
SCHEMBL1825545 0.80 KMT2A (0.43) KMT2AMEN1TSHRDHODH
SCHEMBL1823194 0.80 KMT2A (0.43) KMT2AMEN1TSHRDHODH
SCHEMBL1823816 0.79 KMT2A (0.44) KMT2AKDRBRAF
SCHEMBL1823818 0.79 KMT2A (0.44) KMT2AKDRBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118051-A1 NEW COMPOUNDS, METHODS FOR THEIR PREPARATION AND USE THEREOF Chelsea Therapeutics, Inc. (US) 2009-11-18 EP disclosed
WO-2008097180-A1 NEW COMPOUNDS, METHODS FOR THEIR PREPARATION AND USE THEREOF CHELSEA THERAPEUTICS, INC. (US) 2008-08-14 WO disclosed