SCHEMBL4448190

SCHEMBL4448190

CCCCC[n+]1ccn(CCCOC(=O)[C@](O)(c2ccccc2)[C@@H]2CCCC(F)(F)C2)c1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.45
ALDH1A1 P00352 2/20 0.41
CHRM2 P08172 12/20 0.40
CHRM1 P11229 12/20 0.40
SLC6A3 Q01959 2/20 0.40
KCNH2 Q12809 2/20 0.40
POLB P06746 1/20 0.40
CHRM3 P20309 11/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP2C19 P33261 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
PKM P14618 1/20 0.38
NFKB1 P19838 1/20 0.38
THPO P40225 1/20 0.38
ABCB11 O95342 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL2796363 0.99 HTT (0.45) HTTALDH1A1CHRM2CHRM1SLC6A3
Bromide SCHEMBL3676930 0.99 HTT (0.45) HTTALDH1A1CHRM2CHRM1SLC6A3
Bromide SCHEMBL3679014 0.97 HTT (0.45) HTTALDH1A1CHRM2CHRM1SLC6A3
Bromide SCHEMBL2794178 0.97 HTT (0.45) HTTALDH1A1CHRM2CHRM1SLC6A3
Bromide SCHEMBL2795785 0.95 HTT (0.42) HTTALDH1A1CHRM2CHRM1SLC6A3
Bromide SCHEMBL2797746 0.95 HTT (0.46) HTTALDH1A1CHRM2CHRM1SLC6A3
Bromide SCHEMBL2794159 0.95 HTT (0.42) HTTCHRM2CHRM1CHRM3
Bromide SCHEMBL2792719 0.95 HTT (0.46) HTTALDH1A1CHRM2CHRM1SLC6A3
Bromide SCHEMBL2792073 0.93 HTT (0.42) HTTALDH1A1CHRM2CHRM1SLC6A3
Bromide SCHEMBL2792277 0.92 HTT (0.43) HTTCHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2111861-A1 Compositions of phosphodiesterase type IV inhibitors Ranbaxy Laboratories Limited (IN) 2009-10-28 EP claimed
EP-2111861-A1 Compositions of phosphodiesterase type IV inhibitors Ranbaxy Laboratories Limited (IN) 2009-10-28 EP disclosed