SCHEMBL4448425

SCHEMBL4448425

CCOc1ccccc1CNS(=O)(=O)c1cccc2c(NC(C)=O)cccc12

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.46
POLB P06746 2/20 0.46
MAPT P10636 2/20 0.46
TSHR P16473 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.46
ALOX12 P18054 1/20 0.46
EDNRA P25101 1/20 0.44
GAA P10253 1/20 0.44
CCR8 P51685 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4452477 0.89 MEN1 (0.48) TP53POLBMAPTEDNRAGAA
SCHEMBL4448161 0.83 NPY5R (0.50) POLBEDNRACCR8MEN1KMT2A
SCHEMBL4449069 0.83 EDNRA (0.51) POLBALDH1A1HPGDEDNRAGAA
SCHEMBL4449293 0.83 MEN1 (0.45) ALDH1A1EDNRACCR8MEN1KMT2A
SCHEMBL4622884 0.82 NSD2 (0.52) EDNRACCR8KMT2A
SCHEMBL4447174 0.82 KDM4E (0.51) ALDH1A1EDNRACCR8KMT2ALMNA
SCHEMBL4448268 0.82 MCL1 (0.55) TP53POLBMAPTTSHRALDH1A1
SCHEMBL4448820 0.81 EDNRA (0.49) EDNRACCR8KMT2A
SCHEMBL4445783 0.81 NSD2 (0.60) POLBMAPTTSHRALDH1A1HPGD
SCHEMBL4448991 0.80 NAMPT (0.46) POLBEDNRACCR8MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547716-B2 Sulfonamide derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. (JP) 2009-06-16 US disclosed
EP-1402890-B1 SULFONAMIDE DERIVATIVES INST MED MOLECULAR DESIGN INC (JP) 2008-01-09 EP disclosed
US-20040234622-A1 Sulfonamide derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. (JP) 2004-11-25 US disclosed
EP-1402890-A1 SULFONAMIDE DERIVATIVES Institute of Medicinal Molecular Design, Inc. (JP) 2004-03-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040234622-A1 Sulfonamide derivatives PCNA, TOP2A, DDB1 TP53 52/4885POLB 56/4885MAPT 4821/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.