Bromide

Bromide

SCHEMBL4449437

CC(C)c1nc(Cl)nc(-c2ccc(F)cc2)c1C[P+](c1ccccc1)(c1ccccc1)c1ccccc1.[Br-]

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GCGR P47871 16/20 0.41
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
GLA P06280 1/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4449474 0.79 GCGR (0.63) GCGR
SCHEMBL27885298 0.79 GCGR (0.49) GCGR
Bromide SCHEMBL426277 0.78 JAK1 (0.36) GCGR
Bromide SCHEMBL426278 0.78 AKT1 (0.52) ALDH1A1
SCHEMBL4455298 0.78 GCGR (0.48) GCGR
SCHEMBL2347107 0.74 GCGR (0.42) GCGR
SCHEMBL4462472 0.73 GCGR (0.48) GCGRKDM4EALDH1A1
SCHEMBL27885299 0.72 GCGR (0.39) GCGR
Trifluoromethanesulfonic Acid SCHEMBL17967550 0.72 AKT1 (0.49) ALDH1A1
SCHEMBL2344461 0.72 GCGR (0.40) GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009157014-A2 A PROCESS FOR PREPARING HMG-COA REDUCTASE INHIBITORS AND INTERMEDIATES CADILA HEALTHCARE LIMITED (IN) 2009-12-30 WO claimed
WO-2009157014-A2 A PROCESS FOR PREPARING HMG-COA REDUCTASE INHIBITORS AND INTERMEDIATES CADILA HEALTHCARE LIMITED (IN) 2009-12-30 WO disclosed