SCHEMBL4449706

SCHEMBL4449706

COc1cc(NC(=O)O)ccc1-n1ccnc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.65
CYP19A1 P11511 1/20 0.52
CYP11B1 P15538 1/20 0.52
CYP11B2 P19099 1/20 0.52
PSEN1 P49768 2/20 0.47
PSEN2 P49810 2/20 0.47
APH1B Q8WW43 2/20 0.47
NCSTN Q92542 2/20 0.47
APH1A Q96BI3 2/20 0.47
PSENEN Q9NZ42 2/20 0.47
QPCT Q16769 1/20 0.46
CD38 P28907 2/20 0.45
GRM4 Q14833 1/20 0.44
POLB P06746 1/20 0.44
HTT P42858 1/20 0.44
CYP3A4 P08684 1/20 0.43
ABL1 P00519 1/20 0.43
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1038335 0.83 AAK1 (0.61) AAK1CYP19A1CYP11B1CYP11B2PSEN1
SCHEMBL3312814 0.81 CYP19A1 (0.55) AAK1CYP19A1CYP11B1CYP11B2POLB
SCHEMBL4456548 0.81 PSEN1 (0.64) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL17783138 0.80 AAK1 (1.00) AAK1
SCHEMBL3316441 0.80 KMT2A (0.56) AAK1POLBHTTKDM4ENPC1
SCHEMBL16388652 0.80 AAK1 (1.00) AAK1
SCHEMBL9290092 0.79 CYP11B1 (0.61) AAK1CYP19A1CYP11B1CYP11B2PSEN1
SCHEMBL3313160 0.78 AAK1 (0.53) AAK1CYP19A1CYP11B1CYP11B2PSEN1
SCHEMBL27159848 0.77 CYP11B1 (0.60) AAK1CYP19A1CYP11B1CYP11B2PSEN1
SCHEMBL3313965 0.77 AAK1 (0.55) AAK1CYP19A1CYP11B1CYP11B2QPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2019093-A1 UREA TYPE CINNAMIDE DERIVATIVE Eisai R&D Management Co., Ltd. (JP) 2009-01-28 EP disclosed