SCHEMBL4451573

SCHEMBL4451573

c1ccc(-c2cccc(P(c3cccc(-c4ccccc4)c3)c3cccc(-c4ccccc4)c3)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.55
TDP1 Q9NUW8 1/20 0.55
MAOA P21397 1/20 0.48
ALDH1A1 P00352 3/20 0.47
MGLL Q99685 3/20 0.43
ESR1 P03372 3/20 0.42
ESR2 Q92731 2/20 0.42
HDAC8 Q9BY41 2/20 0.41
KMO O15229 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC2 Q92769 1/20 0.41
ALOX5 P09917 1/20 0.41
PRSS1 P07477 1/20 0.40
PRSS2 P07478 1/20 0.40
PRSS3 P35030 1/20 0.40
AGXT P21549 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP2C9 P11712 1/20 0.39
HSD17B1 P14061 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27456368 0.97 CYP3A4 (0.60) CYP3A4TDP1MAOAALDH1A1MGLL
Hydrochloric Acid SCHEMBL5433165 0.97 CYP3A4 (0.52) CYP3A4TDP1MAOAALDH1A1MGLL
SCHEMBL13572520 0.93 CYP3A4 (0.55) CYP3A4TDP1MAOAALDH1A1MGLL
SCHEMBL22101140 0.84 CYP3A4 (0.44) CYP3A4TDP1MAOAALDH1A1MGLL
SCHEMBL19480054 0.84 CYP3A4 (0.44) CYP3A4TDP1MAOAALDH1A1MGLL
Biphenyl SCHEMBL6633071 0.83 CYP3A4 (0.80) CYP3A4TDP1MAOAALDH1A1ESR1
Biphenyl SCHEMBL4383765 0.80 CYP3A4 (0.75) CYP3A4TDP1MAOAALDH1A1ESR1
SCHEMBL15698273 0.80 TDP1 (0.75) CYP3A4TDP1MAOAALDH1A1ESR1
SCHEMBL1314228 0.80 TDP1 (0.75) CYP3A4TDP1MAOAALDH1A1ESR1
Biphenyl SCHEMBL4381705 0.80 CYP3A4 (0.75) CYP3A4TDP1MAOAALDH1A1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8648000-B2 Diene polymerisation INEOS COMMERCIAL SERVICES UK LIMITED (GB) 2014-02-11 US claimed
WO-2012035546-A3 A TAMPER EVIDENT MULTIPLE METALLIZED AND DEMETALLIZED SECURITY DEVICE AND PROCESS FOR PREPARING THE SAME KAPOOR AJAY (IN) 2012-05-10 WO claimed
EP-1918312-B1 Diene polymerisation INEOS COMMERCIAL SERVICES UK (GB) 2011-12-07 EP claimed
US-20080293896-A1 Diene polymerisation INEOS SALES (UK) LIMITED (GB) 2008-11-27 US claimed
EP-1918312-A1 Diene polymerisation INEOS EUROPE LIMITED (GB) 2008-05-07 EP claimed
US-20020137820-A1 Phosphorus compounds SANDOZ LTD. (CH) 2002-09-26 US claimed
US-4182813-A CATALYST COMPRISING A COBALT COMPOUND, ORGANOALUMINUM COMPOUND, AND AN ORGANIC PHOSPHORUS COMPOUND JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1980-01-08 US claimed
EP-3702404-B1 POLYMER COMPOSITION AND TIRE ENEOS MAT CORPORATION (JP) 2024-07-17 EP disclosed
EP-3702404-A1 POLYMER COMPOSITION AND TIRE JSR Corporation (JP) 2020-09-02 EP disclosed
US-8648000-B2 Diene polymerisation INEOS COMMERCIAL SERVICES UK LIMITED (GB) 2014-02-11 US disclosed
WO-2012035546-A3 A TAMPER EVIDENT MULTIPLE METALLIZED AND DEMETALLIZED SECURITY DEVICE AND PROCESS FOR PREPARING THE SAME KAPOOR AJAY (IN) 2012-05-10 WO disclosed
EP-1918312-B1 Diene polymerisation INEOS COMMERCIAL SERVICES UK (GB) 2011-12-07 EP disclosed
US-7579057-B2 Resin molding and worked item therefrom JSR CORPORATION (JP) 2009-08-25 US disclosed
US-5879805-A USING CATALYST COMPRISING A COBALT COMPOUND, A PHOSPHINE, XANTHOGEN THIOCYANIDE, CARBON DISULFIDE, AN ORGANOALUMINUM COMPOUND UNION CARBIDE CHEMICALS & PLASTICS TECHNOLOGY CORPORATION (US) 1999-03-09 US disclosed
US-5548045-A USING A COORDINATION CATALYST COMPOSED OF A COBALT COMPOUND, ORGANOALUMINUM COMPOUND AND A PHOSPHINE COMPOUND JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1996-08-20 US disclosed
US-5488079-A HEAT AND LIGHT STABILIZERS FOR OLEFINS USING PHOSPHINES SANDOZ LTD. (CH) 1996-01-30 US disclosed
EP-0511015-A1 Process for producing polybutadiene JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1992-10-28 EP disclosed
US-4255543-A LOW MOLECULAR WEIGHT POLYMER USING A CATALYST COMPRISING A COBALT COMPOUND, AN ORGANIC PHOSPHINE, A TRIALKYL ALUMINUM COMPOUND, AND AN ALKYLALUMINUM HALIDE JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1981-03-10 US disclosed
US-4182813-A CATALYST COMPRISING A COBALT COMPOUND, ORGANOALUMINUM COMPOUND, AND AN ORGANIC PHOSPHORUS COMPOUND JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1980-01-08 US disclosed
US-4176219-A COORDINATION CATALYST OF A COBALT AND PHOSPHINE COMPOUND, A TRIALKYLALUMINUM, WATER AND A HYDROCARBYL HALIDE JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1979-11-27 US disclosed