SCHEMBL4452605

SCHEMBL4452605

CN(C)C1CCC(c2cnc3c(c2)C(c2cnn(CCN4CCOCC4)c2)CN3)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.35
MAPK8 P45983 2/20 0.34
MAPK9 P45984 2/20 0.34
MAPK10 P53779 2/20 0.34
HRH3 Q9Y5N1 3/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
KCNH2 Q12809 1/20 0.33
MAPK1 P28482 1/20 0.33
HDAC4 P56524 1/20 0.33
EZH2 Q15910 4/20 0.32
TBK1 Q9UHD2 3/20 0.32
SLC6A4 P31645 2/20 0.32
IKBKE Q14164 2/20 0.32
NRAS P01111 1/20 0.32
FLT3 P36888 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
PIK3CD O00329 1/20 0.32
KDM5B Q9UGL1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10227428 0.84 GSK3B (0.32) MAPK8MAPK9MAPK10HRH3CYP3A4
SCHEMBL4471248 0.78 MAPK8 (0.53) MAPK8MAPK9MAPK10HRH3CYP3A4
SCHEMBL2753042 0.74 MAPK8 (0.63) MAPK8MAPK9MAPK10MAPK1PIK3CD
SCHEMBL2753263 0.74 MAPK8 (0.63) MAPK8MAPK9MAPK10MAPK1PIK3CD
SCHEMBL4457547 0.69 MAPK8 (0.30) MAPK8MAPK9MAPK10
SCHEMBL4458450 0.67 MAPK8 (0.39) MAPK8MAPK9MAPK10HRH3KDM5B
SCHEMBL2752645 0.66 PIK3CD (0.43) MAP4K4MAPK8MAPK9MAPK10HRH3
SCHEMBL4457793 0.66 GSK3B (0.40) MAPK8MAPK9MAPK10HRH3CYP2C9
SCHEMBL4465305 0.66 MAPK8 (0.36) MAPK8MAPK9MAPK10IRAK4
SCHEMBL14027119 0.65 SLC6A4 (0.32) SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178552-B2 7-Azaindole derivatives and their use in the inhibition of c-Jun N-terminal kinase EISAI R&D MANAGEMENT CO., LTD. (JP) 2012-05-15 US disclosed