SCHEMBL4452782

SCHEMBL4452782

CC(N)CC1COCCO1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.47
CHRM4 P08173 1/20 0.47
CHRM5 P08912 1/20 0.47
CHRM3 P20309 1/20 0.47
ALDH1A1 P00352 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
RAB9A P51151 1/20 0.30
THRB P10828 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13745062 1.00 CHRM2 (0.47) CHRM2CHRM4CHRM5CHRM3ALDH1A1
SCHEMBL104458 0.83 CHRM2 (0.50) CHRM2CHRM4CHRM5CHRM3ALDH1A1
SCHEMBL20793588 0.83 CHRM2 (0.50) CHRM2CHRM4CHRM5CHRM3ALDH1A1
SCHEMBL20793890 0.83 CHRM2 (0.50) CHRM2CHRM4CHRM5CHRM3ALDH1A1
SCHEMBL28397337 0.82
SCHEMBL23250876 0.81 CHRM2 (0.48) CHRM2CHRM4CHRM5CHRM3ALDH1A1
SCHEMBL23250875 0.81 CHRM2 (0.48) CHRM2CHRM4CHRM5CHRM3ALDH1A1
SCHEMBL11928865 0.81 CHRM2 (0.48) CHRM2CHRM4CHRM5CHRM3ALDH1A1
Hydrochloric Acid SCHEMBL30673767 0.80
SCHEMBL8895315 0.79 CHRM2 (0.47) CHRM2CHRM4CHRM5CHRM3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819000-B1 NODULISPORIC ACID DERIVATIVES MERCK & CO INC (US) 2009-07-08 EP disclosed
EP-0819000-A4 NODULISPORIC ACID DERIVATIVES MERCK & CO INC (US) 2001-04-11 EP disclosed
EP-0986552-A1 5-NAPHTHALEN-1-YL-1,3-DIOXANE DERIVATIVES, PREPARATION AND THERAPEUTIC APPLICATION SANOFI-SYNTHELABO (FR) 2000-03-22 EP disclosed
US-5962499-A ACARICIDAL, ANTIPARASITIC, INSECTICIDAL AND ANTHELMINTIC AGENTS MERCK & CO., INC. (US) 1999-10-05 US disclosed
WO-1998055474-A1 5-NAPHTHALEN-1-YL-1,3-DIOXANE DERIVATIVES, PREPARATION AND THERAPEUTIC APPLICATION SANOFI-SYNTHELABO (FR) 1998-12-10 WO disclosed
EP-0819000-A1 NODULISPORIC ACID DERIVATIVES Merck & Co., Inc. (US) 1998-01-21 EP disclosed
WO-1996029073-A1 NODULISPORIC ACID DERIVATIVES MERCK & CO., INC. (US) 1996-09-26 WO disclosed