SCHEMBL4453830

SCHEMBL4453830

CCCS(=O)(=O)c1ccccc1Nc1nc(Nc2cc(CC=O)c(C)cc2OC(C)C)ncc1Cl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 19/20 0.55
INSR P06213 18/20 0.55
KCNH2 Q12809 2/20 0.52
ZAP70 P43403 2/20 0.52
PLK4 O00444 1/20 0.52
BUB1B O60566 1/20 0.52
JAK2 O60674 1/20 0.52
ROCK2 O75116 1/20 0.52
ABL1 P00519 1/20 0.52
EGFR P00533 1/20 0.52
NTRK1 P04629 1/20 0.52
LCK P06239 1/20 0.52
NPM1 P06748 1/20 0.52
FES P07332 1/20 0.52
LYN P07948 1/20 0.52
RET P07949 1/20 0.52
IGF1R P08069 1/20 0.52
ABCB1 P08183 1/20 0.52
MET P08581 1/20 0.52
ROS1 P08922 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4453827 0.90 ALK (0.68) ALKINSRKCNH2ZAP70PLK4
SCHEMBL1546094 0.87 ZAP70 (0.56) ALKINSRKCNH2ZAP70PLK4
SCHEMBL30165735 0.80 ALK (0.83) ALKINSR
SCHEMBL25566208 0.80 ALK (0.83) ALKINSR
SCHEMBL24853245 0.80 ALK (0.76) ALKINSRKCNH2ZAP70PLK4
SCHEMBL1546454 0.80 ALK (0.82) ALKINSRKCNH2ZAP70PLK4
SCHEMBL1545649 0.77 ALK (0.84) ALKINSRKCNH2
SCHEMBL1546175 0.76 ALK (0.60) ALKINSRKCNH2ZAP70FGFR2
SCHEMBL1546092 0.76 ALK (0.67) ALKINSRKCNH2ZAP70PLK4
SCHEMBL1013964 0.75 ALK (0.69) ALKINSRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091918-A2 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2009-08-26 EP disclosed
WO-2008073687-A2 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2008-06-19 WO disclosed