SCHEMBL4454926

SCHEMBL4454926

COc1cncc2nc[nH]c(=O)c12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 1/20 0.44
KDM4B O94953 1/20 0.44
KDM5C P41229 1/20 0.44
KDM4C Q9H3R0 1/20 0.44
KDM5B Q9UGL1 1/20 0.44
KDM3A Q9Y4C1 1/20 0.44
PARP1 P09874 7/20 0.42
SRC P12931 2/20 0.42
KMT2A Q03164 1/20 0.40
EGFR P00533 1/20 0.40
PDPK1 O15530 4/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
HPGD P15428 2/20 0.37
ADORA3 P0DMS8 1/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
RAB9A P51151 1/20 0.37
SIRT5 Q9NXA8 1/20 0.37
CA12 O43570 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20187523 0.77 PARP1 (0.59) KDM4AKDM4BKDM5CKDM4CKDM5B
SCHEMBL3051495 0.77 PARP1 (0.63) PARP1SRCKMT2AEGFRPDPK1
SCHEMBL29609262 0.75 PDE3B (0.50) PARP1SRCKMT2APDPK1SMN1; SMN2
SCHEMBL615784 0.75 PDE3B (0.50) PARP1SRCKMT2APDPK1SMN1; SMN2
Hydrochloric Acid SCHEMBL15711283 0.75 PARP1 (0.61) PARP1SRCKMT2AEGFRPDPK1
SCHEMBL31204498 0.74 CHEK1 (0.44) PARP1SRCKMT2AEGFRPDPK1
SCHEMBL15710544 0.74 PARP1 (0.44) PARP1SRCKMT2AEGFRPDPK1
SCHEMBL30353912 0.74 PARP1 (0.44) PARP1SRCKMT2AEGFRPDPK1
SCHEMBL17164000 0.74 KDM4A (0.47) KDM4AKDM4BKDM5CKDM4CKDM5B
Hydrochloric Acid SCHEMBL28100847 0.73 PARP1 (0.43) PARP1SRCKMT2AEGFRPDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009154870-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2009-12-23 WO disclosed
WO-2009154870-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2009-12-23 WO disclosed