SCHEMBL4460766

SCHEMBL4460766

CC#CCn1c(NC[C@H](C)NC(=O)OC(C)(C)C)nc2c1c(=O)n(Cc1ccccc1C#N)c(=O)n2C

nearest known ligand 0.48

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 17/20 0.48
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4475888 0.86 DPP4 (0.47) DPP4KMT2A
SCHEMBL4468325 0.84 KMT2A (0.52) DPP4KMT2A
SCHEMBL4468320 0.84 KMT2A (0.52) DPP4KMT2A
SCHEMBL4247782 0.84 DPP4 (0.49) DPP4
SCHEMBL4247777 0.84 DPP4 (0.49) DPP4
SCHEMBL4483700 0.83 DPP4 (0.51) DPP4
SCHEMBL4485715 0.83 DPP4 (0.51) DPP4
SCHEMBL4487738 0.82 DPP4 (0.55) DPP4
SCHEMBL4474941 0.82 DPP4 (0.55) DPP4
SCHEMBL4468010 0.79 DPP4 (0.48) DPP4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7495002-B2 3-methyl-7-butinyl-xanthines, the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-02-24 US disclosed
US-20060079541-A1 3-methyl-7-butinyl-xanthines, the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-04-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060079541-A1 3-methyl-7-butinyl-xanthines, the preparation thereof and their use as pharmaceutical compositions DPP4, DPP7, DPP3 DPP4 1/4885KMT2A 2557/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.