SCHEMBL4460957

SCHEMBL4460957

COc1cccc(C(=O)N2CCC(Oc3ccc(Nc4ncnc5cc(OC)c(OC)cc45)cc3)CC2)c1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.62
ERBB2 P04626 5/20 0.62
KDR P35968 3/20 0.59
ABCB1 P08183 1/20 0.56
ABCG2 Q9UNQ0 1/20 0.56
MAPK7 Q13164 1/20 0.56
LCK P06239 1/20 0.56
RET P07949 1/20 0.56
SRC P12931 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4460085 0.91 ERBB2 (0.70) EGFRERBB2
SCHEMBL4463315 0.84 ERBB2 (0.72) EGFRERBB2
SCHEMBL4458822 0.83 ERBB2 (0.73) EGFRERBB2
SCHEMBL4468336 0.80 ERBB2 (0.70) EGFRERBB2
SCHEMBL3432391 0.80 EGFR (0.88) EGFRERBB2
SCHEMBL4470019 0.79 ERBB2 (0.57) EGFRERBB2KDRRETSRC
SCHEMBL4467463 0.78 ERBB2 (0.73) ERBB2
SCHEMBL16075707 0.77 EGFR (1.00) EGFRERBB2
SCHEMBL4466009 0.76 ERBB2 (0.79) EGFRERBB2
SCHEMBL3395684 0.76 EGFR (0.85) EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7585869-B2 Substituted heterocylces for the treatment of abnormal cell growth PFIZER, INC. (US) 2009-09-08 US claimed