SCHEMBL4467272

SCHEMBL4467272

CSc1ccc(CC(=O)N[C@@H](Cc2cc(F)cc(F)c2)[C@H](O)CNC(C)c2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
BACE1 P56817 10/20 0.47
BCHE P06276 1/20 0.46
CTSD P07339 1/20 0.46
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
KMT2A Q03164 1/20 0.44
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3492292 0.86 BACE1 (0.41) BACE1CTSDHTT
SCHEMBL3492290 0.86 BACE1 (0.41) BACE1CTSDHTT
SCHEMBL3490665 0.85 BACE1 (0.54) BACE1BCHECTSD
SCHEMBL3490666 0.85 BACE1 (0.54) BACE1BCHECTSD
SCHEMBL3491085 0.84 BACE1 (0.40) BACE1CTSD
SCHEMBL3491089 0.84 BACE1 (0.40) BACE1CTSD
SCHEMBL3491446 0.79 BACE1 (0.50) BACE1CTSD
SCHEMBL3491449 0.79 BACE1 (0.50) BACE1CTSD
SCHEMBL3493091 0.79 BACE1 (0.43) BACE1CTSD
SCHEMBL3493086 0.79 BACE1 (0.43) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7589094-B2 N- (3-amino-2-hydroxy-propyl) substituted alkylamide compounds ELAN PHARMACEUTICALS, INC. (US) 2009-09-15 US claimed