SCHEMBL4474425

SCHEMBL4474425

CCN(NCc1ccc(O)c(OC)c1)C(=O)c1cccc(NC(=O)CCN2CCC(OC(=O)N(c3ccccc3-c3ccccc3)c3ccccc3-c3ccccc3)CC2)c1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 20/20 0.46
ADRB2 P07550 19/20 0.46
CHRM2 P08172 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3175566 0.92 CHRM3 (0.54) CHRM3ADRB2CHRM2
SCHEMBL4484440 0.87 CHRM3 (0.40) CHRM3ADRB2
SCHEMBL4494456 0.81 CHRM3 (0.38) CHRM3ADRB2CHRM2
SCHEMBL5801465 0.81 MEN1 (0.34) CHRM3ADRB2
SCHEMBL4474416 0.81 CHRM3 (0.46) CHRM3ADRB2
SCHEMBL4471889 0.81 CHRM3 (0.49) CHRM3ADRB2CHRM2
SCHEMBL4493974 0.80 CHRM3 (0.38) CHRM3ADRB2CHRM2
SCHEMBL3196137 0.79 CHRM3 (0.49) CHRM3ADRB2CHRM2
SCHEMBL4476501 0.78 CHRM2 (0.49) CHRM3ADRB2CHRM2
SCHEMBL265094 0.78 CHRM3 (0.57) CHRM3ADRB2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632847-B2 Bronchodilators; treating chronic obstructive pulmonary disease or asthma; long duration of action; reduced side effects, such as dry-mouth and constipation; e.g. biphenyl-2-ylcarbamic acid 1-(2-(3-[3-(4-hydroxybenzylamino)propionylamino]benzoylamino)ethyl)piperidin-4-yl ester THERAVANCE, INC. (US) 2009-12-15 US disclosed