SCHEMBL4479468

SCHEMBL4479468

CCOc1cc(C(CC([NH])=O)N2C(=O)c3ccccc3C2=O)ccc1OC

nearest known ligand 0.82

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 12/20 0.82
PDE4B Q07343 12/20 0.82
PDE4C Q08493 12/20 0.82
PDE4D Q08499 12/20 0.82
TNF P01375 10/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21215174 0.91 PDE4A (0.85) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL6098481 0.90 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL6554664 0.90 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL9977590 0.90 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL3120500 0.90 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL6966344 0.90 PDE4A (0.67) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL7746632 0.89 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL6098976 0.87 PDE4A (0.81) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL537314 0.87 PDE4A (0.81) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL4927794 0.86 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DTNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1605935-A4 METHODS OF USING AND COMPOSITIONS COMPRISING SELECTIVE CYTOKINE INHIBITORY DRUGS FOR THE TREATMENT AND MANAGEMENT OF DISORDERS OF THE CENTRAL NERVOUS SYSTEM CELGENE CORP (US) 2009-05-20 EP disclosed
EP-1605935-A2 METHODS OF USING AND COMPOSITIONS COMPRISING SELECTIVE CYTOKINE INHIBITORY DRUGS FOR THE TREATMENT AND MANAGEMENT OF DISORDERS OF THE CENTRAL NERVOUS SYSTEM CELGENE CORPORATION (US) 2005-12-21 EP disclosed
WO-2004080393-A2 SELECTIVE CYTOKINE INHIBITORY DRUGS FOR TREATING DISORDERS OF THE CENTRAL NERVOUS SYSTEM CELGENE CORPORATION (US) 2004-09-23 WO disclosed