SCHEMBL4479635

SCHEMBL4479635

COc1cc2c(Oc3ccc(Nc4ccc(C(C)(C)C)cc4)cc3)ccnc2cc1OCCCN1CCC(N2CCCCC2)CC1

nearest known ligand 0.87

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 15/20 0.87
KIT P10721 2/20 0.60
PDGFRA P16234 2/20 0.60
KDR P35968 2/20 0.60
PDGFRB P09619 1/20 0.60
HRH3 Q9Y5N1 1/20 0.56
MET P08581 2/20 0.50
AXL P30530 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4468988 0.99 FGFR2 (0.85) FGFR2KITPDGFRAKDRPDGFRB
SCHEMBL4466866 0.96 FGFR2 (0.80) FGFR2KITPDGFRAKDRPDGFRB
SCHEMBL4486327 0.95 FGFR2 (0.80) FGFR2KITPDGFRAKDRPDGFRB
SCHEMBL4471592 0.93 FGFR2 (1.00) FGFR2KITPDGFRAKDRPDGFRB
SCHEMBL4478491 0.93 FGFR2 (1.00) FGFR2KITPDGFRAKDRPDGFRB
SCHEMBL4479490 0.92 FGFR2 (0.98) FGFR2KITPDGFRAKDRPDGFRB
SCHEMBL4487243 0.91 FGFR2 (0.95) FGFR2KITPDGFRAKDRPDGFRB
SCHEMBL4464922 0.90 FGFR2 (0.82) FGFR2KITPDGFRAKDRPDGFRB
SCHEMBL4482503 0.89 FGFR2 (0.92) FGFR2KITPDGFRAKDRPDGFRB
SCHEMBL4480969 0.89 FGFR2 (0.92) FGFR2KITPDGFRAKDRPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7495104-B2 Quinoline or quinazoline derivatives inhibiting auto-phosphorylation of fibroblast growth factor receptors KIRIN BEER KABUSHIKI KAISHA (JP) 2009-02-24 US claimed
US-7495104-B2 Quinoline or quinazoline derivatives inhibiting auto-phosphorylation of fibroblast growth factor receptors KIRIN BEER KABUSHIKI KAISHA (JP) 2009-02-24 US disclosed
US-7495104-B2 Quinoline or quinazoline derivatives inhibiting auto-phosphorylation of fibroblast growth factor receptors KIRIN BEER KABUSHIKI KAISHA (JP) 2009-02-24 US disclosed
EP-1447405-A1 QUINOLINE OR QUINAZOLINE DERIVATIVES INHIBITING AUTO-PHOSPHORYLATION OF FIBROBLAST GROWTH FACTOR RECEPTORS KIRIN BEER KABUSHIKI KAISHA (JP) 2004-08-18 EP disclosed