SCHEMBL4481935

SCHEMBL4481935

CN(CCN1CCC(OC(=O)N(c2ccccc2-c2ccccc2)N(C(=O)O)c2ccccc2-c2ccccc2)CC1)C(=O)c1cccc(NC(=O)CN2CCNC(=O)C2)c1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.42
ALDH1A1 P00352 2/20 0.39
POLB P06746 1/20 0.39
CHRM3 P20309 13/20 0.39
ADRB2 P07550 5/20 0.39
SMN1; SMN2 Q16637 2/20 0.36
TRPV4 Q9HBA0 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34
DRD4 P21917 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4481938 0.94 CHRM2 (0.45) CHRM2ALDH1A1POLBCHRM3ADRB2
SCHEMBL4495584 0.89 CHRM2 (0.45) CHRM2ALDH1A1POLBCHRM3ADRB2
SCHEMBL4493982 0.89 CHRM2 (0.45) CHRM2ALDH1A1CHRM3ADRB2SMN1; SMN2
SCHEMBL265424 0.88 CHRM2 (0.56) CHRM2CHRM3ADRB2
SCHEMBL4483376 0.86 CHRM2 (0.46) CHRM2CHRM3ADRB2
SCHEMBL4485665 0.85 CHRM2 (0.45) CHRM2CHRM3ADRB2
SCHEMBL4466758 0.85 CHRM2 (0.45) CHRM2CHRM3ADRB2
SCHEMBL4476500 0.85 CHRM2 (0.45) CHRM2ALDH1A1POLBCHRM3ADRB2
SCHEMBL4489639 0.85 CHRM2 (0.45) CHRM2CHRM3ADRB2
SCHEMBL4471155 0.85 CHRM2 (0.45) CHRM2ALDH1A1CHRM3ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632847-B2 Bronchodilators; treating chronic obstructive pulmonary disease or asthma; long duration of action; reduced side effects, such as dry-mouth and constipation; e.g. biphenyl-2-ylcarbamic acid 1-(2-(3-[3-(4-hydroxybenzylamino)propionylamino]benzoylamino)ethyl)piperidin-4-yl ester THERAVANCE, INC. (US) 2009-12-15 US disclosed