SCHEMBL4484665

SCHEMBL4484665

O=C(O)C(O)Cc1nc2ccccc2o1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.54
NPC1 O15118 5/20 0.54
MAPT P10636 2/20 0.54
SMN1; SMN2 Q16637 4/20 0.50
TP53 P04637 2/20 0.50
LMNA P02545 1/20 0.50
LOXL2 Q9Y4K0 1/20 0.49
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.45
PTPRA P18433 1/20 0.44
HPGD P15428 2/20 0.43
AKR1B1 P15121 2/20 0.43
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
GFER P55789 2/20 0.43
HTT P42858 1/20 0.43
ELANE P08246 1/20 0.43
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7909117 0.87 NPC1 (0.58) RAB9ANPC1MAPTSMN1; SMN2TP53
SCHEMBL5288034 0.83 NPC1 (0.53) RAB9ANPC1MAPTSMN1; SMN2TP53
SCHEMBL1627274 0.83 NPC1 (0.53) RAB9ANPC1MAPTSMN1; SMN2TP53
SCHEMBL11099516 0.83 NPC1 (0.53) RAB9ANPC1MAPTSMN1; SMN2TP53
SCHEMBL3112570 0.77 NPC1 (0.61) RAB9ANPC1MAPTSMN1; SMN2TP53
SCHEMBL31614347 0.77 NPC1 (0.61) RAB9ANPC1MAPTSMN1; SMN2TP53
SCHEMBL28737938 0.76 NPC1 (0.56) RAB9ANPC1MAPTSMN1; SMN2TP53
SCHEMBL11360212 0.76 NPC1 (0.47) RAB9ANPC1MAPTSMN1; SMN2TP53
Water SCHEMBL21626175 0.76 NPC1 (0.59) RAB9ANPC1MAPTSMN1; SMN2TP53
SCHEMBL5535419 0.75 MAPT (0.63) RAB9ANPC1MAPTSMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7576198-B1 Integrase inhibitors containing aromatic heterocycle derivatives SHIONOGI & CO., LTD. (JP) 2009-08-18 US disclosed
EP-1219607-A1 INTEGRASE INHIBITORS CONTAINING AROMATIC HETEROCYCLE DERIVATIVES SHIONOGI & CO., LTD. (JP) 2002-07-03 EP disclosed