SCHEMBL448551

SCHEMBL448551

C1=CCc2c(ccc3c4c(ccc23)=CC=C4)=C1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3204886 0.77
SCHEMBL14941252 0.77
SCHEMBL9938341 0.76
SCHEMBL15903546 0.73
SCHEMBL29564692 0.73
SCHEMBL15903796 0.72
SCHEMBL7631751 0.71
SCHEMBL670186 0.71 KDM4E (0.31)
SCHEMBL9287611 0.70
SCHEMBL15903667 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 366 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240358898-A1 Drug Delivery System for Medical Devices RONTIS HELLAS S.A. (GR) 2024-10-31 US claimed
EP-4340823-A1 DRUG DELIVERY SYSTEM FOR MEDICAL DEVICES Rontis Hellas S.A. (GR) 2024-03-27 EP claimed
WO-2022223090-A1 DRUG DELIVERY SYSTEM FOR MEDICAL DEVICES RONTIS HELLAS S.A. (GR) 2022-10-27 WO claimed
EP-3268314-A2 METHOD FOR THE REMOVAL OF ORGANIC CONTAMINANTS FROM WATER Avore NV (BE) 2018-01-17 EP claimed
WO-2016142443-A2 METHOD FOR THE REMOVAL OF ORGANIC CONTAMINANTS FROM WATER AVORE NV (BE) 2016-09-15 WO claimed
EP-2167481-B1 METHOD FOR PRODUCING PROPYLENE OXIDE SUMITOMO CHEMICAL CO (JP) 2011-10-12 EP claimed
US-7999125-B2 Method for producing propylene oxide SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2011-08-16 US claimed
US-20100197945-A1 METHOD FOR PRODUCING PROPYLENE OXIDE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2010-08-05 US claimed
US-20080206161-A1 QUIESCENT FOAMABLE COMPOSITIONS, STEROIDS, KITS AND USES THEREOF FOAMIX PHARMACEUTICALS LTD. (IL) 2008-08-28 US claimed
EP-1890679-A2 STEROID KIT AND FOAMABLE COMPOSITION AND USES THEREOF Foamix Ltd. (IL) 2008-02-27 EP claimed
WO-2007012977-A2 STEROID KIT AND FOAMABLE COMPOSITION AND USES THEREOF FOAMIX LTD (US) 2007-02-01 WO claimed
US-20060264408-A1 Sod minic multifunctional compounds for treating inflammatory bowel disease YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2006-11-23 US claimed
US-20060247216-A1 Steroid compounds comprising superoxide dismutase mimic groups and nitric oxide donor groups, and their use in the preparation of medicaments YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2006-11-02 US claimed
US-20060018937-A1 Steroid kit and foamable composition and uses thereof FOAMIX LTD. 2006-01-26 US claimed
EP-1603556-A2 SOD MIMIC MULTIFUNCTIONAL COMPOUNDS FOR TREATING INFLAMMATORY BOWEL DISEASE YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2005-12-14 EP claimed
EP-1562975-A2 STEROID COMPOUNDS COMPRISING SUPEROXIDE DISMUTASE MIMIC GROUPS AND NITRIC OXIDE DONOR GROUPS, AND THEIR USE IN THE PREPARATION OF MEDICAMENTS YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2005-08-17 EP claimed
WO-2004078172-A2 SOD MIMIC MULTIFUNCTIONAL COMPOUNDS FOR TREATING INFLAMMATORY BOWEL DISEASE YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2004-09-16 WO claimed
WO-2004037843-A2 STEROID COMPOUNDS COMPRISING SUPEROXIDE DISMUTASE MIMIC GROUPS AND NITRIC OXIDE DONOR GROUPS, AND THEIR USE IN THE PREPARATION OF MEDICAMENTS YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2004-05-06 WO claimed
EP-0973791-A2 PROCESS FOR PREPARATION OF 7 ALPHA-CARBOXYL 9, 11-EPOXY STEROIDS AND INTERMEDIATES USEFUL THEREIN AND A GENERAL PROCESS FOR THE EPOXIDATION OF OLIFINIC DOUBLE BONDS G.D. Searle &amp; Co. (US) 2000-01-26 EP claimed
WO-1997021720-A2 PROCESSES FOR PREPARATION OF 7 ALPHA-CARBOXYL 9,11-EPOXY STEROIDS AND INTERMEDIATES USEFUL THEREIN AND A GENERAL PROCESS FOR THE EPOXIDATION OF OLIFINIC DOUBLE BONDS G.D. SEARLE AND CO. (US) 1997-06-19 WO claimed