SCHEMBL4485671

SCHEMBL4485671

O=C(CNC1CC1)Nc1cccc(C(=O)CNCCN2CCC(OC(=O)N(c3ccccc3-c3ccccc3)c3ccccc3-c3ccccc3)CC2)c1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 18/20 0.41
CARM1 Q86X55 1/20 0.41
PRMT6 Q96LA8 1/20 0.41
HTR1A P08908 1/20 0.40
HTR7 P34969 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4475972 0.94 CHRM3 (0.40) CHRM3CARM1PRMT6HTR1AHTR7
SCHEMBL4490236 0.93 CHRM3 (0.43) CHRM3CARM1PRMT6
SCHEMBL4471158 0.92 CHRM3 (0.42) CHRM3CARM1PRMT6
SCHEMBL4466761 0.92 CHRM3 (0.45) CHRM3CARM1PRMT6
SCHEMBL264834 0.89 CHRM3 (0.55) CHRM3
SCHEMBL4493985 0.89 CHRM3 (0.41) CHRM3CARM1PRMT6
SCHEMBL4478187 0.88 CHRM3 (0.40) CHRM3CARM1PRMT6
SCHEMBL4476551 0.88 CHRM3 (0.43) CHRM3CARM1PRMT6
SCHEMBL4478362 0.85 CHRM3 (0.42) CHRM3CARM1PRMT6
SCHEMBL4494146 0.85 EPHX2 (0.46) CHRM3CARM1PRMT6HTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632847-B2 Bronchodilators; treating chronic obstructive pulmonary disease or asthma; long duration of action; reduced side effects, such as dry-mouth and constipation; e.g. biphenyl-2-ylcarbamic acid 1-(2-(3-[3-(4-hydroxybenzylamino)propionylamino]benzoylamino)ethyl)piperidin-4-yl ester THERAVANCE, INC. (US) 2009-12-15 US disclosed