SCHEMBL4489170

SCHEMBL4489170

O=C(Nc1n[nH]c2cc(-c3cccc(F)c3)ccc12)c1ccc(F)cc1F

nearest known ligand 0.66

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 5/20 0.66
GSK3A P49840 2/20 0.66
HDAC6 Q9UBN7 7/20 0.54
CYP1A2 P05177 1/20 0.53
FGFR1 P11362 2/20 0.52
FGFR2 P21802 2/20 0.52
FGFR3 P22607 2/20 0.52
FGFR4 P22455 3/20 0.51
AAK1 Q2M2I8 1/20 0.50
CDKL2 Q92772 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4483422 0.93 HDAC6 (0.62) GSK3BGSK3AHDAC6CYP1A2FGFR1
SCHEMBL4493662 0.92 GSK3B (0.63) GSK3BGSK3AHDAC6CYP1A2FGFR1
SCHEMBL4494622 0.92 HDAC6 (0.65) GSK3BGSK3AHDAC6FGFR1FGFR2
SCHEMBL4503270 0.92 GSK3B (0.56) GSK3BGSK3AHDAC6CYP1A2FGFR1
SCHEMBL4488592 0.91 GSK3B (0.66) GSK3BGSK3AHDAC6CYP1A2FGFR1
SCHEMBL4492586 0.90 GSK3B (0.58) GSK3BGSK3AHDAC6CYP1A2FGFR1
SCHEMBL4480650 0.90 GSK3B (0.54) GSK3BGSK3AHDAC6CYP1A2FGFR1
SCHEMBL4489400 0.89 GSK3B (0.53) GSK3BGSK3AHDAC6CYP1A2FGFR1
SCHEMBL4494611 0.89 HDAC6 (0.67) GSK3BGSK3AHDAC6FGFR1FGFR2
SCHEMBL4484175 0.87 HDAC6 (0.52) GSK3BGSK3AHDAC6CYP1A2FGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632854-B2 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them PFIZER ITALIA S.R.L. (IT) 2009-12-15 US claimed