SCHEMBL4491840

SCHEMBL4491840

CCOc1ccccc1-c1ccc2c(NC(=O)c3cccc(Cl)c3)n[nH]c2c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 6/20 0.62
FGFR1 P11362 5/20 0.62
FGFR3 P22607 5/20 0.62
HDAC6 Q9UBN7 11/20 0.60
FGFR4 P22455 3/20 0.57
GSK3B P49841 2/20 0.54
HDAC1 Q13547 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
CDC7 O00311 1/20 0.49
DAPK3 O43293 1/20 0.49
PAK4 O96013 1/20 0.49
CDK2 P24941 1/20 0.49
FLT3 P36888 1/20 0.49
CSNK1A1 P48729 1/20 0.49
CLK2 P49760 1/20 0.49
CDK7 P50613 1/20 0.49
CDK9 P50750 1/20 0.49
PRKX P51817 1/20 0.49
CDK5 Q00535 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4492073 0.89 FGFR1 (0.62) FGFR2FGFR1FGFR3HDAC6FGFR4
SCHEMBL4486822 0.87 HDAC6 (0.62) FGFR2FGFR1FGFR3HDAC6FGFR4
SCHEMBL4493253 0.87 FGFR2 (0.60) FGFR2FGFR1FGFR3HDAC6FGFR4
SCHEMBL4497949 0.86 GSK3B (0.55) FGFR2FGFR1FGFR3HDAC6FGFR4
SCHEMBL4493689 0.85 HDAC6 (0.62) FGFR2FGFR1FGFR3HDAC6FGFR4
SCHEMBL4495202 0.84 HDAC6 (0.68) FGFR2FGFR1FGFR3HDAC6FGFR4
SCHEMBL4483037 0.83 HDAC6 (0.58) FGFR2FGFR1FGFR3HDAC6GSK3B
SCHEMBL4477062 0.83 HDAC6 (0.57) FGFR2FGFR1FGFR3HDAC6FGFR4
SCHEMBL4504172 0.83 GSK3B (0.56) FGFR2FGFR1FGFR3HDAC6FGFR4
SCHEMBL4486923 0.83 HDAC6 (0.73) FGFR2FGFR1FGFR3HDAC6FGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632854-B2 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them PFIZER ITALIA S.R.L. (IT) 2009-12-15 US claimed