SCHEMBL4495586

SCHEMBL4495586

CN(CCN1CCC(OC(=O)N(c2ccccc2-c2ccccc2)c2ccccc2-c2ccccc2)CC1)C(=O)c1cccc(NC(=O)CN2CCCC2)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.49
HPGD P15428 1/20 0.44
CHRM3 P20309 11/20 0.43
ADRB2 P07550 1/20 0.41
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
DRD4 P21917 2/20 0.41
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4476501 0.94 CHRM2 (0.49) CHRM2CHRM3ADRB2POLBSMN1; SMN2
SCHEMBL4495584 0.93 CHRM2 (0.45) CHRM2HPGDCHRM3ADRB2POLB
SCHEMBL265208 0.90 CHRM2 (0.61) CHRM2CHRM3
SCHEMBL4483379 0.90 CHRM2 (0.49) CHRM2CHRM3ADRB2
SCHEMBL4489644 0.89 CHRM2 (0.48) CHRM2CHRM3ADRB2
SCHEMBL4481938 0.89 CHRM2 (0.45) CHRM2CHRM3ADRB2POLBSMN1; SMN2
SCHEMBL4493982 0.88 CHRM2 (0.45) CHRM2CHRM3ADRB2SMN1; SMN2ALDH1A1
SCHEMBL4476500 0.87 CHRM2 (0.45) CHRM2CHRM3ADRB2POLBSMN1; SMN2
SCHEMBL4486950 0.86 EPHX2 (0.46) HPGDCHRM3POLBSMN1; SMN2ALDH1A1
SCHEMBL266402 0.85 CHRM2 (0.60) CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632847-B2 Bronchodilators; treating chronic obstructive pulmonary disease or asthma; long duration of action; reduced side effects, such as dry-mouth and constipation; e.g. biphenyl-2-ylcarbamic acid 1-(2-(3-[3-(4-hydroxybenzylamino)propionylamino]benzoylamino)ethyl)piperidin-4-yl ester THERAVANCE, INC. (US) 2009-12-15 US disclosed