SCHEMBL4497815

SCHEMBL4497815

Nc1nc(Nc2ccc(N3CCCC(O)C3)cc2)sc1C(=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 10/20 0.52
CCND1 P24385 10/20 0.52
CDK11A Q9UQ88 9/20 0.51
CCNT1 O60563 8/20 0.51
CDK9 P50750 8/20 0.51
CDK6 Q00534 8/20 0.51
CDK5 Q00535 4/20 0.51
LTK P29376 1/20 0.51
CLK2 P49760 1/20 0.51
GSK3A P49840 1/20 0.51
GSK3B P49841 1/20 0.51
CDK7 P50613 1/20 0.51
LIMK1 P53667 1/20 0.51
PRKCQ Q04759 1/20 0.51
TAOK1 Q7L7X3 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
ALK Q9UM73 1/20 0.51
CDK5R1 Q15078 3/20 0.47
CCNA2 P20248 3/20 0.47
CDK2 P24941 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4333612 0.91 CDK4 (0.51) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4343119 0.85 CDK4 (0.56) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4333379 0.84 CDK4 (0.56) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL5745076 0.83 CDK4 (0.74) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4338443 0.83 CDK4 (0.56) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4331535 0.82 CDK5 (0.47) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4336027 0.81 CDK4 (0.54) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4331555 0.79 CDK4 (0.51) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4342717 0.79 CDK4 (0.57) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4335185 0.79 CDK4 (0.55) CDK4CCND1CDK11ACCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740576-B1 NOVEL PIPERIDINE SUBSTITUTED DIAMINOTHIAZOLES HOFFMANN LA ROCHE (CH) 2009-07-01 EP disclosed