SCHEMBL4500326

SCHEMBL4500326

CCN(CC)Cc1nc(Nc2ccccc2)sc1C(=O)NCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD O00767 2/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
LMNA P02545 2/20 0.47
ALOX12 P18054 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
NPC1 O15118 7/20 0.46
RAB9A P51151 7/20 0.46
MAPT P10636 6/20 0.46
HPGD P15428 3/20 0.46
ALDH1A1 P00352 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
DHODH Q02127 1/20 0.43
GAA P10253 1/20 0.43
POLB P06746 1/20 0.43
CDK2 P24941 2/20 0.42
CDC7 O00311 1/20 0.42
CCNE1 P24864 1/20 0.42
DBF4 Q9UBU7 1/20 0.42
CDK5 Q00535 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580738 0.86 SCD (0.52) SCDMEN1KMT2ALMNANPSR1
SCHEMBL3584381 0.83 CHRM4 (0.48) SCDLMNANPSR1HPGDALDH1A1
SCHEMBL3592976 0.83 SCD (0.49) SCDMEN1KMT2ALMNANPSR1
SCHEMBL5364912 0.77 KMT2A (0.67) SCDMEN1KMT2ALMNAALOX12
SCHEMBL4929895 0.73 SCD (0.64) SCDMEN1KMT2ALMNANPSR1
SCHEMBL5365211 0.72 CDC7 (0.55) SCDMEN1KMT2ALMNAALOX12
SCHEMBL5369173 0.71 KMT2A (0.59) MEN1KMT2ALMNAALOX12NPSR1
SCHEMBL5397042 0.70 KMT2A (0.58) MEN1KMT2ALMNAALOX12NPSR1
SCHEMBL4398547 0.70 NPC1 (0.53) MEN1KMT2ALMNAALOX12NPSR1
SCHEMBL3593166 0.69 SCD (0.55) SCDMEN1KMT2ALMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029138-A1 AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2009-03-04 EP disclosed
WO-2007130075-A1 AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2007-11-15 WO disclosed