SCHEMBL4519703

SCHEMBL4519703

CC(=O)c1cnc(N)s1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL4610612 0.98 TSHR (0.46)
SCHEMBL1636287 0.80
SCHEMBL1631557 0.80
Water SCHEMBL28159942 0.78 HCAR2 (0.55)
Hydrochloric Acid SCHEMBL1984729 0.78 HCAR2 (0.55)
SCHEMBL27582970 0.78
SCHEMBL21469422 0.78
SCHEMBL4219879 0.78 HDAC1 (0.50)
SCHEMBL5875612 0.78
SCHEMBL23224219 0.78 SMN1; SMN2 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 85 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12365657-B2 Preparation of 2-chloro-1-(2-chlorothiazol-5-yl)ethanone BASF SE (DE) 2025-07-22 US claimed
CN-114555568-B Preparation of 2-chloro-1- (2-chlorothiazol-5-yl) ethanone 巴斯夫欧洲公司 2025-01-24 CN claimed
US-20240051929-A1 PREPARATION OF 2-CHLORO-1-(2-CHLOROTHIAZOL-5-YL)ETHANONE BASF SE (DE) 2024-02-15 US claimed
EP-4038056-B1 PREPARATION OF 2-CHLORO-1-(2-CHLOROTHIAZOL-5-YL)ETHANONE BASF SE (DE) 2023-11-08 EP claimed
CN-114555568-A Preparation of 2-chloro-1- (2-chlorothiazol-5-yl) ethanone 巴斯夫欧洲公司 2022-05-27 CN claimed
WO-2021063880-A1 PREPARATION OF 2-CHLORO-1-(2-CHLOROTHIAZOL-5-YL)ETHANONE BASF SE (DE) 2021-04-08 WO claimed
JP-2006504796-A 2006-02-09 JP claimed
EP-1551815-A1 THIAZOLE COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS Pfizer Products Inc. (US) 2005-07-13 EP claimed
US-20040152747-A1 Thiazole compounds for treatment of neurodegenerative disorders PFIZER INC 2004-08-05 US claimed
WO-2004033439-A1 THIAZOLE COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS PFIZER PRODUCTS INC. (US) 2004-04-22 WO claimed
US-12365657-B2 Preparation of 2-chloro-1-(2-chlorothiazol-5-yl)ethanone BASF SE (DE) 2025-07-22 US disclosed
CN-112739695-B Novel thiazole derivative and pharmaceutically acceptable salt thereof 永进药品工业株式会社 2025-03-18 CN disclosed
CN-114555568-B Preparation of 2-chloro-1- (2-chlorothiazol-5-yl) ethanone 巴斯夫欧洲公司 2025-01-24 CN disclosed
US-12110299-B2 Thiazole derivatives and pharmaceutically acceptable salts thereof YUNGJIN PHARM. CO., LTD. (KR) 2024-10-08 US disclosed
CN-118666863-A Pyrimidothienothiazole derivative or pharmaceutically acceptable salt thereof, and preparation and application thereof 皖南医学院 2024-09-20 CN disclosed
WO-2004033439-A1 THIAZOLE COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS PFIZER PRODUCTS INC. (US) 2004-04-22 WO disclosed
US-4104268-A POLYACRYLONITRILE, POLYESTERS, POLYAMIDES BAYER AKTIENGESELLSCHAFT (DE) 1978-08-01 US disclosed
US-4058617-A BACTERICIDES, AMOBICIDES, SCHISTOSOMES, FILARIAE, TRICHOMONADES CIBA-GEIGY CORPORATION (US) 1977-11-15 US disclosed
US-4006127-A Cationic diazacyanine dyestuffs BAYER AKTIENGESELLSCHAFT (DT) 1977-02-01 US disclosed
US-3998952-A AMOEBICIDES, BACTERICIDES, FUNGICIDES CIBA-GEIGY CORPORATION (US) 1976-12-21 US disclosed