SCHEMBL4531330

SCHEMBL4531330

O=c1c2c(Cl)cccc2ncn1C1CCCNC1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 11/20 0.45
HTR6 P50406 4/20 0.44
PIK3R2 O00459 4/20 0.40
PRKCI P41743 1/20 0.39
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
HTR2B P41595 1/20 0.39
HTR3A P46098 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
PIM1 P11309 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
PARP1 P09874 1/20 0.38
CNR1 P21554 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16587068 0.83 CLK1 (0.46) PARP1CNR1
SCHEMBL16333800 0.80 ACVR1 (0.51) HTR6PRKCI
SCHEMBL23518636 0.80 ACVR1 (0.51) HTR6PRKCI
SCHEMBL16333798 0.80 ACVR1 (0.51) HTR6PRKCI
SCHEMBL30417848 0.76 IDO1 (0.43) PIK3CDPIK3R2PARP1CNR1
SCHEMBL30418923 0.73 IDO1 (0.43) PIK3CDPIK3R2PARP1CNR1
SCHEMBL30419567 0.73 HSD17B13 (0.47) PIK3CDPIK3R2PARP1
SCHEMBL283372 0.71 CRBN (0.64)
SCHEMBL16382725 0.71 KDM4E (0.48) HTR6PRKCIHTR2BPARP1
SCHEMBL18945874 0.71 CRBN (0.64)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7635700-B2 e.g. 3-(5-METHYL-4-OXO-4H-QUINAZOLIN-3-YL)-PIPERIDINE-2,6-DIONE; cytokine (epidermal/fibroblast/endothelial/tumor necrosis growth factors) antagonist; antitumor, antiinflammatory agent, neurodegenerative diseases CELGENE CORPORATION (US) 2009-12-22 US disclosed