SCHEMBL4540063

SCHEMBL4540063

CNS(=O)(=O)C(C)c1ccc2[nH]cc(C3CCN(C)CC3)c2c1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 12/20 0.60
HTR1B P28222 12/20 0.60
HTR1A P08908 2/20 0.60
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
CYP2C9 P11712 1/20 0.59
THPO P40225 1/20 0.59
HTR1F P30939 1/20 0.54
APP P05067 1/20 0.54
MAPT P10636 1/20 0.53
BLM P54132 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HTR6 P50406 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9875206 0.89 HTR1D (0.60) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL252679 0.81 HTR1D (0.60) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL8915192 0.80 CYP1A2 (0.68) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL8416068 0.76 HTR1D (0.62) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL3260325 0.75 HTR1D (0.59) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL3260327 0.75 HTR1D (0.59) HTR1DHTR1BHTR1ACYP1A2CYP3A4
Naratriptan SCHEMBL68753 0.75 HTR1D (1.00) HTR1DHTR1BHTR1ACYP1A2CYP3A4
Naratriptan SCHEMBL29403931 0.75 HTR1D (1.00) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL3546728 0.75 CYP1A2 (1.00) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL30908918 0.75 CYP1A2 (1.00) HTR1DHTR1BHTR1ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009118753-A2 PROCESS FOR PREPARATION OF NARATRIPTAN HYDROCHLORIDE USV LIMITED (IN) 2009-10-01 WO claimed