SCHEMBL4549632

SCHEMBL4549632

N/N=C\N(N)c1ccc(CC(=O)N2CCN(CCc3ccc4nonc4c3)CC2)cn1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 15/20 0.53
KCNH2 Q12809 13/20 0.53
SIGMAR1 Q99720 1/20 0.38
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
ECE2 P0DPD6 1/20 0.35
SLC6A4 P31645 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15196934 0.75 KCNJ1 (0.63) KCNJ1KCNH2SLC6A4
SCHEMBL15196712 0.75 KCNJ1 (0.79) KCNJ1KCNH2SLC6A4
SCHEMBL2731338 0.72 KCNH2 (0.76) KCNJ1KCNH2SIGMAR1
SCHEMBL15196767 0.70 KCNJ1 (0.75) KCNJ1KCNH2SLC6A4
SCHEMBL15196781 0.70 KCNH2 (0.61) KCNJ1KCNH2SLC6A4
SCHEMBL2731436 0.70 KCNJ1 (1.00) KCNJ1KCNH2SLC6A4
SCHEMBL4549576 0.69 KCNH2 (0.81) KCNJ1KCNH2SLC6A4
SCHEMBL9731780 0.69 KCNH2 (0.71) KCNJ1KCNH2
SCHEMBL15191673 0.67 KCNJ1 (0.91) KCNJ1KCNH2SLC6A4
SCHEMBL297835 0.66 KCNJ1 (0.64) KCNJ1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012058134-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2012-05-03 WO disclosed