SCHEMBL4549643

SCHEMBL4549643

CCC(Cc1ccc2c(c1)COC2=O)N1CCN(C(=O)Cc2ccc(-n3cnnn3)cc2)CC1

nearest known ligand 0.70

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 18/20 0.70
KCNJ1 P48048 12/20 0.70
SLC6A4 P31645 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2729675 0.90 KCNH2 (0.72) KCNH2KCNJ1SLC6A4
Hydrochloric Acid SCHEMBL15192220 0.86 KCNH2 (0.66) KCNH2KCNJ1SLC6A4
SCHEMBL4549136 0.82 KCNH2 (1.00) KCNH2KCNJ1SLC6A4
SCHEMBL4549790 0.81 KCNH2 (0.72) KCNH2KCNJ1SLC6A4
SCHEMBL4549561 0.81 KCNH2 (0.72) KCNH2KCNJ1SLC6A4
SCHEMBL4549791 0.81 KCNH2 (0.72) KCNH2KCNJ1SLC6A4
SCHEMBL4549555 0.80 KCNH2 (0.93) KCNH2KCNJ1SLC6A4
SCHEMBL14785840 0.79 KCNH2 (1.00) KCNH2KCNJ1SLC6A4
SCHEMBL14790700 0.79 KCNH2 (1.00) KCNH2KCNJ1SLC6A4
SCHEMBL14785931 0.78 KCNH2 (1.00) KCNH2KCNJ1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012058134-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2012-05-03 WO disclosed