SCHEMBL4550424

SCHEMBL4550424

CCC(=O)Nc1cc(C(=O)NCc2ccc(OCC(F)F)c(CI)c2)ccn1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.48
MAPT P10636 3/20 0.48
ROS1 P08922 1/20 0.38
ALK Q9UM73 1/20 0.38
HDAC1 Q13547 3/20 0.37
MAPK1 P28482 1/20 0.36
KDM1A O60341 2/20 0.36
PPARG P37231 2/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
PTGES O14684 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
LMNA P02545 1/20 0.36
GSK3A P49840 1/20 0.35
ROCK1 Q13464 1/20 0.35
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2715164 0.89 MAPT (0.47) GSK3BMAPTROS1ALKHDAC1
SCHEMBL2716389 0.89 MAPT (0.47) GSK3BMAPTROS1ALKHDAC1
SCHEMBL2714271 0.88 ROS1 (0.47) GSK3BMAPTROS1ALKHDAC1
SCHEMBL2714487 0.88 MAPT (0.47) GSK3BMAPTROS1ALKHDAC1
SCHEMBL2713374 0.83 GSK3B (0.51) GSK3BMAPTJAK2JAK1TYK2
SCHEMBL2713191 0.82 MAPT (0.46) GSK3BMAPTROS1ALKHDAC1
SCHEMBL2715144 0.81 GSK3B (0.44) GSK3BMAPTALKHDAC1KDM1A
SCHEMBL2715453 0.81 MAPT (0.49) GSK3BMAPTMAPK1JAK2JAK1
SCHEMBL2714796 0.80 MAPT (0.43) GSK3BMAPTALKHDAC1KDM1A
SCHEMBL2717172 0.80 MAPT (0.61) GSK3BMAPTROS1ALKHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012053186-A1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2012-04-26 WO disclosed