SCHEMBL4550692

SCHEMBL4550692

CCN(CC)CCCCNc1ncc2c(n1)N(C1CCCC1)C(=O)N(c1cccc(OC)c1F)C2

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.49
CSF1R P07333 9/20 0.49
FGFR1 P11362 10/20 0.47
FGFR4 P22455 9/20 0.47
FGFR2 P21802 8/20 0.47
FGFR3 P22607 8/20 0.47
FYN P06241 1/20 0.39
PDGFRB P09619 1/20 0.39
PDGFRA P16234 1/20 0.39
PRKACA P17612 1/20 0.39
PRKACG P22612 1/20 0.39
PRKACB P22694 1/20 0.39
MAPK1 P28482 1/20 0.39
KDR P35968 1/20 0.39
EPHB3 P54753 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4406583 0.97 EGFR (0.50) EGFRCSF1RFGFR1FGFR4FGFR2
SCHEMBL4412453 0.94 EGFR (0.43) EGFRCSF1RFGFR1FGFR4FGFR2
SCHEMBL5385405 0.91 EGFR (0.44) EGFRCSF1RFGFR1FGFR4FGFR2
SCHEMBL4398823 0.90 EGFR (0.47) EGFRCSF1RFGFR1FGFR4FGFR2
SCHEMBL4395788 0.89 FGFR4 (0.44) EGFRCSF1RFGFR1FGFR4FGFR2
SCHEMBL4410282 0.88 FGFR1 (0.47) EGFRCSF1RFGFR1FGFR4FGFR2
SCHEMBL4403064 0.88 FGFR4 (0.43) EGFRCSF1RFGFR1FGFR4FGFR2
SCHEMBL4404780 0.87 FGFR1 (0.49) FGFR1FGFR4FGFR2FGFR3
SCHEMBL4401790 0.87 FGFR4 (0.54) EGFRCSF1RFGFR1FGFR4FGFR2
SCHEMBL4406900 0.87 FGFR1 (0.48) FGFR1FGFR4FGFR2FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1549651-B1 PYRIMIDOPYRIMIDONES AS KINASE INHIBITORS WARNER LAMBERT CO (US) 2009-12-23 EP disclosed
US-7196090-B2 Kinase inhibitors WARNER-LAMBERT COMPANY (US) 2007-03-27 US disclosed
WO-2006038112-A1 USE OF KINASE INHIBITORS TO PROMOTE NEOCHONDROGENESIS WARNER-LAMBERT COMPANY LLC (US) 2006-04-13 WO disclosed
EP-1549651-A1 KINASE INHIBITORS Warner-Lambert Company LLC (US) 2005-07-06 EP disclosed
WO-2004011465-A1 KINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-05 WO disclosed
US-20040019210-A1 Kinase inhibitors CHIVIKAS CONNOLLY CLEO J (US) 2004-01-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040019210-A1 Kinase inhibitors CDK2, CDK1, CDK4 EGFR 141/4885CSF1R 900/4885FGFR1 88/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.