SCHEMBL4554555

SCHEMBL4554555

CC(=O)NC1(c2cccc(F)c2)CCN(CCC2(c3cccc(Cl)c3Cl)CN(c3ccccc3)C(=O)CO2)CC1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.46
ALDH1A1 P00352 1/20 0.46
TACR3 P29371 11/20 0.43
TACR1 P25103 3/20 0.40
TACR2 P21452 4/20 0.38
GAA P10253 1/20 0.38
HTT P42858 1/20 0.38
OPRM1 P35372 1/20 0.38
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1382015 0.89 TACR3 (0.50) CYP2C19ALDH1A1TACR3TACR1TACR2
Hydrochloric Acid SCHEMBL3906709 0.88 TACR3 (0.49) CYP2C19ALDH1A1TACR3TACR1TACR2
Fumaric Acid SCHEMBL3896093 0.86 TACR3 (0.51) CYP2C19ALDH1A1TACR3TACR1TACR2
Fumaric Acid SCHEMBL3896097 0.86 TACR3 (0.51) CYP2C19ALDH1A1TACR3TACR1TACR2
SCHEMBL1381888 0.82 TACR1 (0.52) TACR3TACR1TACR2
SCHEMBL1381258 0.81 TACR3 (0.52) TACR3TACR1TACR2
SCHEMBL1381405 0.81 TACR2 (0.50) TACR3TACR1TACR2
SCHEMBL1382630 0.80 TACR2 (0.57) CYP2C19ALDH1A1TACR3TACR1TACR2
SCHEMBL3911078 0.80 TACR3 (0.52) TACR3TACR1TACR2
SCHEMBL3896095 0.79 TACR3 (0.42) CYP2C19ALDH1A1TACR3TACR1TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2131842-A2 USE OF A COMPOUND ANTAGONIST TO THE NK-2-RECEPTORS OF A NEUROKININE FOR THE PREPARATION OF DRUGS USEFUL FOR PREVENTING AND TREATING SEXUAL DYSFUNCTION Sanofi-Aventis (FR) 2009-12-16 EP disclosed
WO-2008110697-A2 USE OF A COMPOUND ANTAGONIST TO THE NK2 RECEPTORS OF A NEUROKININE FOR THE PREPARATION OF DRUGS USEFUL FOR PREVENTING AND TREATING SEXUAL DYSFUNCTION SANOFI-AVENTIS (FR) 2008-09-18 WO disclosed