SCHEMBL4557911

SCHEMBL4557911

CCOCCN(C)CCOc1ccc(CCCNc2cc(OC)c(OC)cc2C2CCc3cc(O)ccc3C2)cc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.47
ESR2 Q92731 2/20 0.47
CYP26A1 O43174 1/20 0.36
DRD2 P14416 3/20 0.36
DRD3 P35462 3/20 0.36
GRIN2B Q13224 2/20 0.35
GRIN1 Q05586 1/20 0.35
BCHE P06276 3/20 0.34
ACHE P22303 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL226755 1.00 ESR1 (0.47) ESR1ESR2CYP26A1DRD2DRD3
SCHEMBL229279 0.93 ESR1 (0.48) ESR1ESR2CYP26A1DRD2DRD3
SCHEMBL228223 0.93 ESR1 (0.48) ESR1ESR2CYP26A1DRD2DRD3
SCHEMBL228544 0.93 ESR1 (0.52) ESR1ESR2CYP26A1DRD2DRD3
SCHEMBL228883 0.92 ESR1 (0.48) ESR1ESR2CYP26A1DRD2DRD3
SCHEMBL229964 0.92 ESR1 (0.48) ESR1ESR2CYP26A1DRD2DRD3
SCHEMBL228519 0.90 ESR1 (0.51) ESR1ESR2CYP26A1DRD2DRD3
SCHEMBL229683 0.90 ESR1 (0.51) ESR1ESR2CYP26A1DRD2DRD3
SCHEMBL229729 0.90 ESR1 (0.40) ESR1ESR2CYP26A1DRD2DRD3
SCHEMBL228403 0.90 ESR1 (0.47) ESR1ESR2CYP26A1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612114-B2 Such as (R)-6-{2-{ethyl[4-(2-ethylaminoethyl)benzyl]amino }-4-methoxyphenyl }-5,6,7,8-tetrahydronaphthalen-2-ol; osteoporosis; breast cancer EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-11-03 US disclosed