SCHEMBL4558619

SCHEMBL4558619

Cc1cc2nc(C(=O)O)ccc2cc1-c1ccc(OCc2c(-c3c(Cl)cccc3Cl)noc2C2CCC2)cc1

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.65
HSD17B13 Q7Z5P4 1/20 0.60
FABP1 P07148 7/20 0.59
CYP1A2 P05177 1/20 0.59
CYP2C9 P11712 1/20 0.59
FABP4 P15090 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006338 0.89 NR1H4 (0.72) NR1H4HSD17B13FABP1CYP1A2CYP2C9
SCHEMBL2003218 0.87 NR1H4 (0.72) NR1H4HSD17B13FABP1CYP1A2CYP2C9
SCHEMBL2001897 0.85 NR1H4 (0.74) NR1H4HSD17B13FABP1CYP1A2CYP2C9
SCHEMBL4340030 0.85 NR1H4 (0.67) NR1H4HSD17B13FABP1CYP1A2CYP2C9
SCHEMBL2001904 0.82 NR1H4 (0.62) NR1H4HSD17B13FABP1CYP1A2CYP2C9
SCHEMBL1998428 0.82 NR1H4 (0.66) NR1H4HSD17B13FABP1CYP1A2CYP2C9
SCHEMBL13335357 0.82 NR1H4 (0.71) NR1H4HSD17B13FABP1FABP4
SCHEMBL2000305 0.81 NR1H4 (0.62) NR1H4HSD17B13FABP1CYP1A2CYP2C9
SCHEMBL23474151 0.79 NR1H4 (0.63) NR1H4HSD17B13FABP1FABP4
SCHEMBL4340034 0.79 NR1H4 (0.59) NR1H4HSD17B13FABP1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079307-A2 FARNESOID X RECEPTOR AGONISTS SmithKline Beecham Corporation (US) 2009-07-22 EP disclosed
WO-2008051942-A2 FARNESOID X RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2008-05-02 WO disclosed