SCHEMBL4560082

SCHEMBL4560082

Cc1cncc(-c2csc([C@@]3(C)CC(=N)N(C)C(=O)C3Sc3ccccc3)c2)c1

nearest known ligand 0.38

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 8/20 0.38
BACE2 Q9Y5Z0 2/20 0.34
CYP2A6 P11509 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4549244 0.89 BACE1 (0.52) BACE1
SCHEMBL4556671 0.83 BACE1 (0.35) BACE1BACE2CYP2A6
SCHEMBL10186854 0.82 BACE1 (0.41) BACE1BACE2CYP2A6
SCHEMBL4549191 0.72 BACE1 (0.47) BACE1
SCHEMBL4559951 0.72 BACE1 (0.36) BACE1BACE2CYP2A6
SCHEMBL12191155 0.71 BACE1 (0.38) BACE1BACE2
SCHEMBL7542498 0.71 BACE1 (0.38) BACE1BACE2
SCHEMBL4549262 0.70 BACE1 (0.58) BACE1
SCHEMBL4556908 0.69 BACE1 (0.46) BACE1BACE2CYP2A6
SCHEMBL4557575 0.68 BACE1 (0.38) BACE1BACE2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8168641-B2 Aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-01 US disclosed