SCHEMBL4565479

SCHEMBL4565479

NCCCCN(Cc1nc2ccccc2[nH]1)C(O)Cc1ccccn1

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 15/20 0.66
CYP2D6 P10635 2/20 0.47
CHRM2 P08172 1/20 0.47
DRD2 P14416 1/20 0.47
OPRM1 P35372 1/20 0.47
KCNH2 Q12809 1/20 0.47
BCHE P06276 1/20 0.43
CYP1A2 P05177 1/20 0.39
CYP2E1 P05181 1/20 0.39
CYP2C8 P10632 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2B6 P20813 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
RAB9A P51151 1/20 0.39
F2 P00734 1/20 0.39
F10 P00742 1/20 0.39
F7 P08709 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12935367 0.80 CXCR4 (0.74) CXCR4CYP2D6CHRM2DRD2OPRM1
SCHEMBL2084833 0.80 CXCR4 (0.74) CXCR4CYP2D6CHRM2DRD2OPRM1
SCHEMBL2084037 0.79 CXCR4 (1.00) CXCR4CYP2D6CHRM2DRD2OPRM1
SCHEMBL12935366 0.78 CXCR4 (0.78) CXCR4CYP2D6CHRM2DRD2OPRM1
SCHEMBL2084710 0.75 CXCR4 (0.73) CXCR4CYP2D6CHRM2DRD2OPRM1
SCHEMBL11858928 0.74 CXCR4 (0.70) CXCR4CYP2D6CHRM2DRD2OPRM1
SCHEMBL12935355 0.72 CXCR4 (0.78) CXCR4CYP2D6CHRM2DRD2OPRM1
SCHEMBL2086783 0.72 CXCR4 (0.60) CXCR4CYP2D6CHRM2DRD2OPRM1
SCHEMBL15778057 0.71 BCHE (0.65) CXCR4CYP2D6DRD2BCHECYP1A2
SCHEMBL12935351 0.71 CXCR4 (0.59) CXCR4CYP2D6CHRM2DRD2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed