SCHEMBL4566485

SCHEMBL4566485

COc1ccc(Cc2ccccc2N(C)c2cc3c(cn2)cc(-c2cc(N)c(F)cc2Cl)c(=O)n3C)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 9/20 0.41
SRC P12931 9/20 0.41
POLB P06746 1/20 0.35
EGFR P00533 1/20 0.34
TP53 P04637 2/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP11B1 P15538 3/20 0.33
CYP11B2 P19099 3/20 0.33
PIK3CA P42336 1/20 0.32
PRKDC P78527 1/20 0.32
LYN P07948 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4566484 0.85 FGFR1 (0.41) FGFR1SRCPOLBEGFRLYN
SCHEMBL5057701 0.84 FGFR1 (0.43) FGFR1SRCEGFR
SCHEMBL4566697 0.77 FGFR1 (0.39) FGFR1SRCEGFRLYN
SCHEMBL5062666 0.76 FGFR1 (0.38) FGFR1SRCEGFRPIK3CAPRKDC
SCHEMBL14999841 0.76 BTK (0.41) SRCLYN
SCHEMBL14999919 0.75 FGFR4 (0.37) FGFR1SRCLYN
SCHEMBL4565918 0.74 FGFR1 (0.37) FGFR1SRCEGFRLYN
SCHEMBL5063032 0.72 FGFR1 (0.45) FGFR1SRCEGFR
SCHEMBL4420929 0.71 SRC (0.50) FGFR1SRCEGFR
SCHEMBL4566352 0.70 FGFR1 (0.61) FGFR1SRCLYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2063897-A2 KINASE INHIBITORS USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES Deciphera Pharmaceuticals, LLC. (US) 2009-06-03 EP disclosed
WO-2008034008-A2 KINASE INHIBITORS USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES DECIPHERA PHARMACEUTICALS, LLC. (US) 2008-03-20 WO disclosed