SCHEMBL4566752

SCHEMBL4566752

COc1ccc(OC)c(Sc2nc(N)nc(-c3cc(OCC(C)=O)c(Cl)cc3Cl)n2)c1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.39
DHFR P00374 5/20 0.38
ADORA3 P0DMS8 1/20 0.36
TYMS P04818 3/20 0.36
EGFR P00533 1/20 0.36
KDR P35968 1/20 0.36
HSP90AA1 P07900 5/20 0.36
HSP90AB1 P08238 5/20 0.36
PTGER3 P43115 1/20 0.34
DCK P27707 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4097120 0.85 HSP90AB1 (0.40) NPC1DHFRTYMSEGFRKDR
SCHEMBL4096143 0.80 NPC1 (0.47) NPC1DHFRTYMSEGFRKDR
SCHEMBL4372093 0.76 GCGR (0.38) NPC1HSP90AA1
SCHEMBL4102760 0.74 HSP90AB1 (0.41) DHFREGFRKDRHSP90AA1HSP90AB1
SCHEMBL13927519 0.72 HSP90AA1 (0.48) DHFRTYMSEGFRKDRHSP90AA1
SCHEMBL4085571 0.72 NPC1 (0.42) NPC1DHFRADORA3TYMSEGFR
SCHEMBL17349607 0.71 HSP90AA1 (0.47) HSP90AA1HSP90AB1
SCHEMBL17349616 0.70 HSP90AA1 (0.56) NPC1HSP90AA1HSP90AB1
SCHEMBL13928062 0.70 HPGD (0.40) NPC1
SCHEMBL14642199 0.69 LRRK2 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2036895-A1 HSP90 INHIBITOR CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-03-18 EP claimed
EP-2036895-A1 HSP90 INHIBITOR CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-03-18 EP disclosed