SCHEMBL4573528

SCHEMBL4573528

COc1ccc(CN2C(=O)CCCC[C@@H]2C=O)cc1

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 18/20 0.58
HCRTR2 O43614 18/20 0.58
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4573689 1.00 HCRTR1 (0.58) HCRTR1HCRTR2MEN1KMT2A
SCHEMBL3682511 0.92 HCRTR2 (0.54) HCRTR1HCRTR2MEN1KMT2A
SCHEMBL6455357 0.92 HCRTR2 (0.54) HCRTR1HCRTR2MEN1KMT2A
SCHEMBL4573105 0.82 HCRTR1 (0.56) HCRTR1HCRTR2KMT2A
SCHEMBL4573101 0.82 HCRTR1 (0.56) HCRTR1HCRTR2KMT2A
SCHEMBL8366845 0.81 HCRTR1 (0.64) HCRTR1HCRTR2
SCHEMBL1965055 0.81 HCRTR1 (0.64) HCRTR1HCRTR2
SCHEMBL4574022 0.80 HCRTR1 (0.57) HCRTR1HCRTR2
SCHEMBL4574026 0.80 HCRTR1 (0.57) HCRTR1HCRTR2
SCHEMBL19382661 0.80 HCRTR1 (0.62) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008031788-A1 AMINOAZEPINE DERIVATIVES AS HIGHLY EFFICIENT INHIBITORS OF THE INDUCIBLE NITRIC OXIDE SYNTHASE NYCOMED GMBH (DE) 2008-03-20 WO disclosed
WO-2008031788-A1 AMINOAZEPINE DERIVATIVES AS HIGHLY EFFICIENT INHIBITORS OF THE INDUCIBLE NITRIC OXIDE SYNTHASE NYCOMED GMBH (DE) 2008-03-20 WO disclosed