(S)-Norduloxetine

(S)-Norduloxetine

SCHEMBL4573573

NCC[C@H](Oc1cccc2ccccc12)c1cccs1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 9/20 1.00
SLC6A4 P31645 9/20 1.00
SLC6A3 Q01959 8/20 1.00
HTR1A P08908 2/20 0.71
MLNR O43193 1/20 0.71
CACNA1F O60840 1/20 0.71
CYP1A2 P05177 1/20 0.71
ADRB1 P08588 1/20 0.71
CYP3A4 P08684 1/20 0.71
GAA P10253 1/20 0.71
CYP2D6 P10635 1/20 0.71
CYP2C9 P11712 1/20 0.71
DRD2 P14416 1/20 0.71
KCNE1 P15382 1/20 0.71
ADRA2B P18089 1/20 0.71
ADRA2C P18825 1/20 0.71
HTR2A P28223 1/20 0.71
HTR2C P28335 1/20 0.71
MC4R P32245 1/20 0.71
CYP2C19 P33261 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
R-Norduloxetine SCHEMBL2634027 1.00 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3HTR1AMLNR
R-Norduloxetine SCHEMBL3268853 0.99 SLC6A2 (0.97) SLC6A2SLC6A4SLC6A3HTR1AMLNR
R-Norduloxetine SCHEMBL3890591 0.93 SLC6A2 (0.86) SLC6A2SLC6A4SLC6A3HTR1AMLNR
SCHEMBL17280843 0.91 SLC6A2 (0.83) SLC6A2SLC6A4SLC6A3HTR1AMLNR
SCHEMBL27847199 0.90 SLC6A2 (0.82) SLC6A2SLC6A4SLC6A3HTR1AMLNR
SCHEMBL27847200 0.90 SLC6A2 (0.82) SLC6A2SLC6A4SLC6A3HTR1AMLNR
SCHEMBL12212180 0.86 SLC6A2 (0.76) SLC6A2SLC6A4SLC6A3HTR1AMLNR
SCHEMBL4563199 0.86 SLC6A2 (0.76) SLC6A2SLC6A4SLC6A3HTR1AMLNR
SCHEMBL20292590 0.85 CACNA2D1 (0.74) SLC6A2SLC6A4SLC6A3HTR1AMLNR
Methylamine SCHEMBL27678263 0.84 SLC6A2 (0.72) SLC6A2SLC6A4SLC6A3HTR1AMLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008081476-A2 PROCESS FOR PREPARING DULOXETINE HYDROCHLORIDE CADILA HEALTHCARE LIMITED (IN) 2008-07-10 WO claimed
EP-2558455-B1 SYNTHESIS OF DULOXETINE AND/OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF KRKA D D NOVO MESTO (SI) 2017-08-09 EP disclosed
US-7928250-B2 Reduction; condensation SYNTHON BV (NL) 2011-04-19 US disclosed
US-20080171887-A1 Process for making duloxetine and related compounds SYNTHON BV (NL) 2008-07-17 US disclosed
WO-2008081476-A2 PROCESS FOR PREPARING DULOXETINE HYDROCHLORIDE CADILA HEALTHCARE LIMITED (IN) 2008-07-10 WO disclosed
WO-2008081476-A2 PROCESS FOR PREPARING DULOXETINE HYDROCHLORIDE CADILA HEALTHCARE LIMITED (IN) 2008-07-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080171887-A1 Process for making duloxetine and related compounds UGT1A10, UGT1A4, UGT1A6 SLC6A2 33/4885SLC6A4 16/4885SLC6A3 52/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.