SCHEMBL4577868

SCHEMBL4577868

COCC(COC)(COC(=O)c1ccccc1)COC(=O)c1ccccc1

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.82
HIF1A Q16665 1/20 0.82
LMNA P02545 2/20 0.53
TDP1 Q9NUW8 4/20 0.53
SLC6A3 Q01959 2/20 0.53
HTR1A P08908 1/20 0.53
CYP2D6 P10635 1/20 0.53
SCN1A P35498 1/20 0.53
SCN5A Q14524 1/20 0.53
SCN2A Q99250 1/20 0.53
SCN3A Q9NY46 1/20 0.53
TSHR P16473 3/20 0.52
KMT2A Q03164 2/20 0.50
SLC6A2 P23975 1/20 0.50
ALDH1A1 P00352 4/20 0.49
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
ADRB2 P07550 2/20 0.45
ADRB1 P08588 2/20 0.45
ADRB3 P13945 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27620 0.91 MAPK1 (1.00) MAPK1HIF1ALMNATDP1SLC6A3
SCHEMBL235921 0.85 MAPK1 (0.81) MAPK1HIF1ALMNATDP1SLC6A3
SCHEMBL9563647 0.85 MAPK1 (0.89) MAPK1HIF1ALMNATDP1SLC6A3
SCHEMBL27794358 0.84 MAPK1 (0.62) MAPK1HIF1ALMNATDP1SLC6A3
SCHEMBL1786754 0.84 MAPK1 (0.79) MAPK1HIF1ALMNATDP1SLC6A3
SCHEMBL9947121 0.84 MAPK1 (0.79) MAPK1HIF1ALMNATDP1SLC6A3
SCHEMBL2333610 0.81 MAPK1 (0.81) MAPK1HIF1ALMNATDP1SLC6A3
SCHEMBL1681317 0.81 MAPK1 (0.81) MAPK1HIF1ALMNATDP1SLC6A3
SCHEMBL4576866 0.81 MAPK1 (0.81) MAPK1HIF1ALMNATDP1SLC6A3
SCHEMBL12227603 0.81 MAPK1 (0.73) MAPK1HIF1ALMNATDP1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1472293-B1 SOLID CATALYST COMPONENT FOR POLYMERIZATION OF OLEFINS, CATALYST COMPRISING THE SAME AND USE THEREOF CHINA PETROLEUM & CHEM CORP (CN) 2017-04-26 EP disclosed
EP-1666505-B1 CATALYST COMPONENTS CATALYSTS FOR OLEFINIC POLYMERIZATION AND THE USE THEREOF CHINA PETROLEUM & CHEMICAL (CN) 2016-03-23 EP disclosed
US-7388061-B2 Solid catalyst component for polymerization of olefins, catalyst comprising the same and use thereof CHINA PETROLEUM & CHEMICAL CORPORATION (CN) 2008-06-17 US disclosed
US-7332455-B2 Catalyst component and catalyst for olefin polymerization as well as use thereof CHINA PETROLEUM & CHEMICAL CORPORATION (CN) 2008-02-19 US disclosed
EP-1472293-A4 SOLID CATALYST COMPONENT FOR POLYMERIZATION OF OLEFINS, CATALYST COMPRISING THE SAME AND USE THEREOF CHINA PETROLEUM & CHEMICAL (CN) 2008-01-16 EP disclosed
EP-1666505-A1 CATALYST COMPONENTS CATALYSTS FOR OLEFINIC POLYMERIZATION AND THE USE THEREOF China Petroleum & Chemical Corporation (CN) 2006-06-07 EP disclosed
US-20050239636-A1 Solid catalyst component for polymerization of olefins, catalyst comprising the same and use thereof CHINA PETROLEUM & CHEMICAL CORPORATION (CN) 2005-10-27 US disclosed
US-20050119427-A1 Catalyst component and catalyst for olefin polymerization as well as use thereof BEIJING RESEARCH INSTITUTE OF CHEMICAL INDUSTRY, CHINA PETROLEUM & CHEMICAL CORPORATION (CN) 2005-06-02 US disclosed
EP-1472293-A1 SOLID CATALYST COMPONENT FOR POLYMERIZATION OF OLEFINS, CATALYST COMPRISING THE SAME AND USE THEREOF China Petroleum & Chemical Corporation (CN) 2004-11-03 EP disclosed
WO-2003068828-A1 SOLID CATALYST COMPONENT FOR POLYMERIZATION OF OLEFINS, CATALYST COMPRISING THE SAME AND USE THEREOF CHINA PETROLEUM & CHEMICAL CORPORATION (CN) 2003-08-21 WO disclosed