SCHEMBL4580276

SCHEMBL4580276

Clc1ccc(CNc2nccc(N3CCOC[C@@H]3c3ccccc3)n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 7/20 0.53
OGA O60502 1/20 0.46
NR3C2 P08235 1/20 0.45
NUDT1 P36639 1/20 0.45
ACHE P22303 3/20 0.44
BACE1 P56817 1/20 0.44
HTT P42858 1/20 0.41
HDAC6 Q9UBN7 3/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC1 Q13547 1/20 0.40
PLK4 O00444 1/20 0.40
LCK P06239 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4580277 1.00 IDH1 (0.53) IDH1OGANR3C2NUDT1ACHE
SCHEMBL4580169 0.87 CCR4 (0.44) IDH1OGANR3C2NUDT1ACHE
SCHEMBL4582206 0.87 CCR4 (0.44) IDH1OGANR3C2NUDT1ACHE
SCHEMBL4582156 0.86 IDH1 (0.46) IDH1OGANR3C2NUDT1ACHE
SCHEMBL4582161 0.86 IDH1 (0.46) IDH1OGANR3C2NUDT1ACHE
SCHEMBL4581003 0.83 IDH1 (0.44) IDH1OGANR3C2NUDT1ACHE
SCHEMBL4581000 0.83 IDH1 (0.44) IDH1OGANR3C2NUDT1ACHE
SCHEMBL4579677 0.82 IDH1 (0.47) IDH1OGANR3C2NUDT1HDAC6
SCHEMBL4579683 0.82 IDH1 (0.47) IDH1OGANR3C2NUDT1HDAC6
SCHEMBL4580965 0.82 IDH1 (0.46) IDH1OGANR3C2NUDT1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7323464-B2 Pyridine and pyrimidine derivatives CELLTECH R&D LIMITED (GB) 2008-01-29 US claimed
US-20050080258-A1 Pyridine and pyrimidine derivatives GENTEX CORPORATION 2005-04-14 US claimed
US-7323464-B2 Pyridine and pyrimidine derivatives CELLTECH R&D LIMITED (GB) 2008-01-29 US disclosed
US-20050080258-A1 Pyridine and pyrimidine derivatives GENTEX CORPORATION 2005-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050080258-A1 Pyridine and pyrimidine derivatives ROR1, MAPK1, IRAK1 IDH1 424/4885OGA 3642/4885NR3C2 787/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.