SCHEMBL4580943

SCHEMBL4580943

O=C1NCCN(c2ccnc(NCc3cc(F)cc(C(F)(F)F)c3)n2)C1c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
IDH1 O75874 5/20 0.41
VNN1 O95497 1/20 0.38
TACR1 P25103 1/20 0.37
GPR52 Q9Y2T5 2/20 0.37
SCN9A Q15858 1/20 0.36
NTRK1 P04629 1/20 0.36
NTRK3 Q16288 1/20 0.36
NTRK2 Q16620 1/20 0.36
CYP3A4 P08684 3/20 0.36
LMNA P02545 2/20 0.36
TSHR P16473 2/20 0.36
KDM4E B2RXH2 1/20 0.36
KDR P35968 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HRH4 Q9H3N8 1/20 0.35
CCNT1 O60563 1/20 0.34
TERT O14746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4583051 0.90 IDH1 (0.44) HDAC1HDAC8HDAC6IDH1KDR
SCHEMBL4582929 0.85 HDAC1 (0.41) HDAC1HDAC8HDAC6IDH1VNN1
SCHEMBL4581890 0.84 IDH1 (0.54) IDH1HRH4MKNK1MKNK2
SCHEMBL4580658 0.81 IDH1 (0.44) HDAC1HDAC8HDAC6IDH1HRH4
SCHEMBL4579971 0.80 KDM4E (0.42) HDAC1HDAC8HDAC6IDH1VNN1
SCHEMBL4582884 0.80 HRH4 (0.43) HDAC1HDAC8HDAC6IDH1HRH4
SCHEMBL4581479 0.80 IDH1 (0.44) HDAC1HDAC8HDAC6IDH1HRH4
SCHEMBL4579658 0.80 IDH1 (0.46) HDAC1HDAC8HDAC6IDH1HRH4
SCHEMBL4580232 0.80 IDH1 (0.46) IDH1CYP3A4HRH4
SCHEMBL4581840 0.79 OGA (0.53) IDH1VNN1LMNAKDM4EMKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7323464-B2 Pyridine and pyrimidine derivatives CELLTECH R&D LIMITED (GB) 2008-01-29 US claimed
US-20050080258-A1 Pyridine and pyrimidine derivatives GENTEX CORPORATION 2005-04-14 US claimed
US-7323464-B2 Pyridine and pyrimidine derivatives CELLTECH R&D LIMITED (GB) 2008-01-29 US disclosed
US-20050080258-A1 Pyridine and pyrimidine derivatives GENTEX CORPORATION 2005-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050080258-A1 Pyridine and pyrimidine derivatives ROR1, MAPK1, IRAK1 HDAC1 481/4885HDAC8 1903/4885HDAC6 2319/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.